SCHEMBL534967

SCHEMBL534967

[c]1cccc2c1c1c3ccccc3c3ccccc3c1c1ccccc21

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
THRB P10828 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2407351 0.85 HPRT1 (0.35) ALDH1A1CYP1A2THRBHPGDHSD17B10
SCHEMBL24104 0.85 HPRT1 (0.35) ALDH1A1CYP1A2THRBHPGDHSD17B10
SCHEMBL4824194 0.85 HPRT1 (0.35) ALDH1A1CYP1A2THRBHPGDHSD17B10
SCHEMBL2409495 0.82 CYP2A6 (0.33) ALDH1A1CYP1A2HSD17B10
SCHEMBL145165 0.81 HPRT1 (0.48) ALDH1A1CYP1A2THRBHPGDHSD17B10
SCHEMBL1333659 0.78 HPRT1 (0.40) ALDH1A1CYP1A2THRBHPGDHSD17B10
SCHEMBL2413265 0.76 HPRT1 (0.36) ALDH1A1CYP1A2THRBHPGDHSD17B10
SCHEMBL534917 0.76 HSD17B10 (0.48) ALDH1A1CYP1A2THRBHPGDHSD17B10
SCHEMBL844969 0.76 HPRT1 (0.46) ALDH1A1CYP1A2THRBHPGDHSD17B10
SCHEMBL844450 0.76 HPRT1 (0.46) ALDH1A1CYP1A2THRBHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 152 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2674418-B1 BISCARBAZOLE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME IDEMITSU KOSAN CO (JP) 2021-01-06 EP claimed
EP-2790239-B1 MATERIAL FOR ORGANIC ELECTROLUMINESCENT ELEMENT AND ORGANIC ELECTROLUMINESCENT ELEMENT IDEMITSU KOSAN CO (JP) 2020-02-05 EP claimed
US-10147889-B2 Biscarbazole derivative and organic electroluminescent element using same IDEMITSU KOSAN CO., LTD. (JP) 2018-12-04 US claimed
US-10147888-B2 Biscarbazole derivative and organic electroluminescent element using same IDEMITSU KOSAN CO., LTD. (JP) 2018-12-04 US claimed
US-RE46974-E1 Organic electroluminescence device IDEMITSU KOSAN CO., LTD. (JP) 2018-07-31 US claimed
US-20180102484-A1 NEW COMPOUND, ORGANIC ELECTROLUMINESCENCE DEVICE MATERIAL, ORGANIC ELECTROLUMINESCENCE DEVICE AND ELECTRONIC DEVICE IDEMITSU KOSAN CO., LTD. (JP) 2018-04-12 US claimed
US-9647220-B2 Organic multicolor light-emitting apparatus SONY CORPORATION (JP) 2017-05-09 US claimed
US-20160276602-A1 ORGANIC MULTICOLOR LIGHT-EMITTING APPARATUS SONY CORPORATION (JP) 2016-09-22 US claimed
US-20160268517-A1 BISCARBAZOLE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME IDEMITSU KOSAN CO., LTD. (JP) 2016-09-15 US claimed
US-9318709-B2 Material for organic electroluminescence device, and organic electroluminescence device using the same IDEMITSU KOSAN CO., LTD. (JP) 2016-04-19 US claimed
US-9306171-B2 Material for organic electroluminescence device and organic electroluminescence device IDEMITSU KOSAN CO., LTD. (JP) 2016-04-05 US claimed
US-20150249219-A1 BISCARBAZOLE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME IDEMITSU KOSAN CO., LTD. (JP) 2015-09-03 US claimed
US-20140048784-A1 BISCARBAZOLE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME IDEMITSU KOSAN CO., LTD. (JP) 2014-02-20 US claimed
US-20140001451-A1 MATERIAL FOR ORGANIC ELECTROLUMINESCENCE DEVICE, AND ORGANIC ELECTROLUMINESCENCE DEVICE USING THE SAME IDEMITSU KOSAN CO., LTD. (JP) 2014-01-02 US claimed
EP-2674418-A1 BISCARBAZOLE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME Idemitsu Kosan Co., Ltd. (JP) 2013-12-18 EP claimed
EP-2602243-A1 MONOAMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME Idemitsu Kosan Co., Ltd. (JP) 2013-06-12 EP claimed
US-20120199820-A1 MONOAMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME IDEMITSU KOSAN CO., LTD. (JP) 2012-08-09 US claimed
US-20240155945-A1 HIGHLY EFFICIENT BLUE FLUORESCENT ORGANIC EMITTER HAVING A HIGH HOMO LEVEL AND AN ORGANIC ELECTROLUMINESCENCE DEVICE COMPRISING THE SAME IDEMITSU KOSAN CO.,LTD. (JP) 2024-05-09 US disclosed
US-20110279020-A1 Biscarbazole Derivative, Material for Organic Electroluminescence Device and Organic Electroluminescence Device Using The Same IDEMITSU KOSAN CO., LTD. 2011-11-17 US disclosed
US-20110278555-A1 BISCARBAZOLE DERIVATIVE, MATERIAL FOR ORGANIC ELECTROLUMINESCENCE DEVICE AND ORGANIC ELECTROLUMINESCENCE DEVICE USING THE SAME IDEMITSU KOSAN CO., LTD. 2011-11-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120199820-A1 MONOAMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME MAOA, ADRA1A, ADRA1D ALDH1A1 102/4885CYP1A2 137/4885THRB 2632/4885
US-20160268517-A1 BISCARBAZOLE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME L1CAM, CCNT1, CCNA1 ALDH1A1 71/4885CYP1A2 51/4885THRB 2817/4885
US-20110278555-A1 BISCARBAZOLE DERIVATIVE, MATERIAL FOR ORGANIC ELECTROLUMINESCENCE DEVICE AND ORGANIC ELECTROLUMINESCENCE DEVICE USING THE SAME UQCRB, OXA1L, HBS1L ALDH1A1 362/4885CYP1A2 170/4885THRB 3657/4885
US-20110279020-A1 Biscarbazole Derivative, Material for Organic Electroluminescence Device and Organic Electroluminescence Device Using The Same UQCRB, OXA1L, HBS1L ALDH1A1 380/4885CYP1A2 132/4885THRB 3886/4885
US-20150249219-A1 BISCARBAZOLE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME L1CAM, CCNT1, CCNA1 ALDH1A1 75/4885CYP1A2 52/4885THRB 2819/4885
US-10147888-B2 Biscarbazole derivative and organic electroluminescent element using same L1CAM, CCNT1, CCNA1 ALDH1A1 71/4885CYP1A2 51/4885THRB 2817/4885
US-20180102484-A1 NEW COMPOUND, ORGANIC ELECTROLUMINESCENCE DEVICE MATERIAL, ORGANIC ELECTROLUMINESCENCE DEVICE AND ELECTRONIC DEVICE CBX8, MLX, HAX1 ALDH1A1 2418/4885CYP1A2 1832/4885THRB 3988/4885
US-10147889-B2 Biscarbazole derivative and organic electroluminescent element using same L1CAM, CCNT1, CCNA1 ALDH1A1 71/4885CYP1A2 51/4885THRB 2817/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.