SCHEMBL5387372

SCHEMBL5387372

CC(=O)c1ccc(S(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.73
LMNA P02545 3/20 0.73
KMT2A Q03164 2/20 0.73
KDM4E B2RXH2 1/20 0.73
MAPK1 P28482 1/20 0.73
CA12 O43570 1/20 0.61
CA9 Q16790 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.59
HTR6 P50406 1/20 0.58
SMN1; SMN2 Q16637 4/20 0.57
HPGD P15428 4/20 0.56
MEN1 O00255 1/20 0.56
ALDH1A1 P00352 3/20 0.56
GAA P10253 2/20 0.56
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
TP53 P04637 1/20 0.52
THRB P10828 1/20 0.52
PRMT1 Q99873 1/20 0.50
PKM P14618 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrogen Sulfide SCHEMBL28084602 0.98 MAPT (0.71) MAPTLMNAKMT2AKDM4EMAPK1
SCHEMBL4027167 0.91 MAPT (0.61) MAPTLMNAKMT2AKDM4EMAPK1
SCHEMBL18364472 0.88 KMT2A (0.58) MAPTLMNAKMT2AKDM4EMAPK1
SCHEMBL10870974 0.86 HPGD (0.77) MAPTLMNAKMT2AKDM4EMAPK1
(Phenylsulfonyl)Benzene SCHEMBL29058880 0.84 HTR6 (0.74) MAPTLMNAKMT2AKDM4EMAPK1
(Phenylsulfonyl)Benzene SCHEMBL2381369 0.84 HTR6 (0.74) MAPTLMNAKMT2AKDM4EMAPK1
SCHEMBL3773485 0.83 GAA (0.67) MAPTLMNAKMT2AKDM4EMAPK1
SCHEMBL7938512 0.83 HSD17B1 (0.63) MAPTLMNAKMT2AKDM4EMAPK1
SCHEMBL165237 0.83 HTR6 (0.64) MAPTLMNAKMT2ACA12CA9
SCHEMBL24360902 0.82 CA12 (0.70) MAPTLMNAKMT2AKDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9650330-B2 Process for the synthesis of aryl sulfones COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2017-05-16 US claimed
US-20160304447-A1 A PROCESS FOR THE SYNTHESIS OF ARYL SULFONES COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2016-10-20 US claimed
WO-2015087352-A1 A PROCESS FOR THE SYNTHESIS OF ARYL SULFONES COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2015-06-18 WO claimed
US-20220204485-A1 STABILIZATION OF AMYLOIDOGENIC IMMUNOGLOBULIN LIGHT CHAINS THE SCRIPPS RESEARCH INSTITUTE 2022-06-30 US disclosed
US-10759765-B2 Heterocyclic carboxylic acid amide ligand and applications thereof in copper catalyzed coupling reaction of aryl halogeno substitute CE PHARM CO., LTD. (CN) 2020-09-01 US disclosed
US-20190127337-A1 HETEROCYCLIC CARBOXYLIC ACID AMIDE LIGAND AND APPLICATIONS THEREOF IN COPPER CATALYZED COUPLING REACTION OF ARYL HALOGENO SUBSTITUTE CE PHARM CO., LTD. (CN) 2019-05-02 US disclosed
WO-2017177979-A1 HETEROCYCLIC CARBOXYLIC ACID AMIDE LIGAND AND APPLICATIONS THEREOF IN COPPER CATALYZED COUPLING REACTION OF ARYL HALOGENO SUBSTITUTE 中国科学院上海有机化学研究所 2017-10-19 WO disclosed
US-9682938-B2 Pyrazolone derivatives as nitroxyl donors CARDIOXYL PHARMACEUTICALS, INC. (US) 2017-06-20 US disclosed
US-9650330-B2 Process for the synthesis of aryl sulfones COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2017-05-16 US disclosed
US-9650330-B2 Process for the synthesis of aryl sulfones COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2017-05-16 US disclosed
US-9650330-B2 Process for the synthesis of aryl sulfones COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2017-05-16 US disclosed
US-5349090-A Process for preparing arylketoamines HOECHST CELANESE CORPORATION (US) 1994-09-20 US disclosed
US-5338884-A Reacting an arylisonitrosoalkanone with hydrogen then acid, ester inpresence of catalyst HOECHST CELANESE (US) 1994-08-16 US disclosed
US-5220063-A Reacting arylisonitrosoalkanone with hydrogen and acyl doner in presence of transition metal catalyst HOECHST CELANESE CORPORATION (US) 1993-06-15 US disclosed
US-5198585-A Catalytic hydrogenation of arylisonitrosoalkanone HOECHST CELANESE CORPORATION (US) 1993-03-30 US disclosed
WO-1993001158-A1 METHOD FOR THE PREPARATION OF ARYLKETOAMINES HOECHST CELANESE CORPORATION (US) 1993-01-21 WO disclosed
US-5175368-A Hydrogenating aryl alpha-oximinoalkyl ketones in aqueous medium containing hydrochlroic acid, recovering salt HOECHST CELANESE CORPORATION (US) 1992-12-29 US disclosed
EP-0491557-A1 Process for the preparation of arylalkylamines and substituted arylalkylamines HOECHST CELANESE CORPORATION (US) 1992-06-24 EP disclosed
US-5041669-A Reacting alkyl aryl ketones with alkyl nitrites, extracting product, catalytically hydrogenating/reducing in nonaqueous acid mixture HOECHST CELANESE CORPORATION (US) 1991-08-20 US disclosed
US-4055652-A 1-[β(R-thio)phenethyl]imidazoles and derivatives thereof SYNTEX (U.S.A.) INC. (US) 1977-10-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220204485-A1 STABILIZATION OF AMYLOIDOGENIC IMMUNOGLOBULIN LIGHT CHAINS TTR, MAP1LC3B, SAAL1 MAPT 41/4885LMNA 478/4885KMT2A 4134/4885
US-20190127337-A1 HETEROCYCLIC CARBOXYLIC ACID AMIDE LIGAND AND APPLICATIONS THEREOF IN COPPER CATALYZED COUPLING REACTION OF ARYL HALOGENO SUBSTITUTE AOC1, AOC2, AOC3 MAPT 4463/4885LMNA 4664/4885KMT2A 1850/4885
US-20160304447-A1 A PROCESS FOR THE SYNTHESIS OF ARYL SULFONES ARSA, TPST2, STS MAPT 2353/4885LMNA 4387/4885KMT2A 806/4885
US-10759765-B2 Heterocyclic carboxylic acid amide ligand and applications thereof in copper catalyzed coupling reaction of aryl halogeno substitute AOC1, AOC2, AOC3 MAPT 4463/4885LMNA 4664/4885KMT2A 1850/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.