SCHEMBL54119

SCHEMBL54119

NC(=O)c1ccccc1B(O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.52
ALDH1A1 P00352 2/20 0.52
MAPT P10636 2/20 0.52
TSHR P16473 2/20 0.52
HSD17B10 Q99714 2/20 0.52
HPGD P15428 1/20 0.52
BCAT2 O15382 1/20 0.52
METAP2 P50579 1/20 0.48
IRAK4 Q9NWZ3 1/20 0.46
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
NPC1 O15118 2/20 0.44
GAA P10253 1/20 0.42
CTNNB1 P35222 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
RAB9A P51151 1/20 0.41
POLB P06746 1/20 0.41
CYP3A4 P08684 1/20 0.41
PARP1 P09874 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29468958 1.00 KDM4E (0.52) KDM4EALDH1A1MAPTTSHRHSD17B10
Alcohol SCHEMBL29246862 0.92 BCAT2 (0.50) KDM4EALDH1A1MAPTTSHRHSD17B10
SCHEMBL25541451 0.82 ENPP2 (0.40) KDM4EALDH1A1MAPTTSHRHSD17B10
SCHEMBL3787789 0.81 BCAT2 (0.42) KDM4EALDH1A1MAPTTSHRHSD17B10
Boric Acid SCHEMBL31026556 0.80 ALDH1A1 (0.61) KDM4EALDH1A1MAPTTSHRHSD17B10
SCHEMBL18919333 0.79 BCAT2 (0.37) KDM4EALDH1A1MAPTTSHRHSD17B10
SCHEMBL29956608 0.79 PARP1 (0.41) KDM4EALDH1A1MAPTTSHRHSD17B10
SCHEMBL519802 0.79 ENPP2 (0.41) KDM4EALDH1A1MAPTPOLBL3MBTL1
SCHEMBL29446522 0.79 ALDH1A1 (0.59) KDM4EALDH1A1MAPTTSHRHSD17B10
SCHEMBL29469063 0.79 ENPP2 (0.41) KDM4EALDH1A1MAPTPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 318 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119081323-A Wear-resistant impact-resistant high polymer floor and preparation process thereof 洁玛新材料股份有限公司 2024-12-06 CN claimed
CN-118063863-A Double-functional nano-particle for rapidly detecting sterilizing bacteria and preparation method and application thereof 江苏省农业科学院 2024-05-24 CN claimed
EP-2718265-B1 PROCESS FOR PREPARING [(3-HYDROXYPYRIDINE-2-CARBONYL)AMINO]ALKANOIC ACIDS, ESTERS AND AMIDES AKEBIA THERAPEUTICS INC (US) 2015-12-16 EP claimed
US-9145366-B2 Process for preparing [(3-hydroxypyridine-2-carbonyl)amino]alkanoic acids, esters and amides AKEBIA THERAPEUTICS, INC. (US) 2015-09-29 US claimed
EP-2718265-A1 PROCESS FOR PREPARING [(3-HYDROXYPYRIDINE-2-CARBONYL)AMINO]ALKANOIC ACIDS, ESTERS AND AMIDES Akebia Therapeutics Inc. (US) 2014-04-16 EP claimed
WO-2012170377-A1 PROCESS FOR PREPARING [(3-HYDROXYPYRIDINE-2-CARBONYL)AMINO]ALKANOIC ACIDS, ESTERS AND AMIDES AKEBIA THERAPEUTICS INC. (US) 2012-12-13 WO claimed
US-20120309977-A1 PROCESS FOR PREPARING [(3-HYDROXYPYRIDINE-2-CARBONYL)AMINO]ALKANOIC ACIDS, ESTERS AND AMIDES AKEBIA THERAPEUTICS INC. (US) 2012-12-06 US claimed
CN-122028918-A TRIM7 inhibitors and uses thereof 沙塔克实验室有限公司 2026-05-12 CN disclosed
EP-4720044-A1 AROMATIC AMIDES AND CONJUGATES THEREOF AS BINDERS TO TEAD Beactica Therapeutics AB (SE) 2026-04-08 EP disclosed
US-12378224-B2 Heteroaryl compounds and their use as Mer inhibitors DONG-A SOCIO HOLDINGS CO., LTD. (KR) 2025-08-05 US disclosed
EP-4069697-B1 CRF RECEPTOR ANTAGONISTS AND METHODS OF USE NEUROCRINE BIOSCIENCES INC (US) 2025-07-16 EP disclosed
WO-2025042797-A1 TRIM7 INHIBITORS AND USES THEREOF SHATTUCK LABS, INC. (US) 2025-02-27 WO disclosed
WO-2025042798-A1 TRIM7 INHIBITORS AND USES THEREOF SHATTUCK LABS, INC. (US) 2025-02-27 WO disclosed
US-20060111375-A1 Compound having tgfß inhibitory activity and medicinal composition containing the same KIRIN BEER KABUSHIKI KAISHA (JP) 2006-05-25 US disclosed
EP-1643998-A1 DUAL NK1/NK3 ANTAGONISTS FOR TREATING SCHIZOPHRENIA F. HOFFMANN-LA ROCHE AG (CH) 2006-04-12 EP disclosed
WO-2005058876-A1 PYRAZINE DERIVATIVES AS EFFECTIVE COMPOUNDS AGAINST INFECTIOUS DISEASES GPC BIOTECH AG (DE) 2005-06-30 WO disclosed
EP-1548008-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND MEDICINAL COMPOSITION CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2005-06-29 EP disclosed
US-20050119347-A1 Microbicidal agents on the basis of biphenyl benzamide derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2005-06-02 US disclosed
US-20050090533-A1 Dual NK1/NK3 receptor antagonists F. HOFMANN-LA ROCHE AG (CH) 2005-04-28 US disclosed
WO-2005002577-A1 DUAL NK1/NK3 ANTAGONISTS FOR TREATING SCHIZOPHRENIA F. HOFFMANN-LA ROCHE AG (CH) 2005-01-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050119347-A1 Microbicidal agents on the basis of biphenyl benzamide derivatives DDT, MSR1, CYP1B1 KDM4E 1352/4885ALDH1A1 169/4885MAPT 4798/4885
US-20060111375-A1 Compound having tgfß inhibitory activity and medicinal composition containing the same TGFB1, TGFBR1, TGFBR2 KDM4E 1176/4885ALDH1A1 1257/4885MAPT 2587/4885
US-20050090533-A1 Dual NK1/NK3 receptor antagonists TACR2, TAC3, TACR1 KDM4E 1504/4885ALDH1A1 1516/4885MAPT 4611/4885
US-12378224-B2 Heteroaryl compounds and their use as Mer inhibitors MERTK, RET, ERBB2 KDM4E 1635/4885ALDH1A1 3864/4885MAPT 1125/4885
US-20120309977-A1 PROCESS FOR PREPARING [(3-HYDROXYPYRIDINE-2-CARBONYL)AMINO]ALKANOIC ACIDS, ESTERS AND AMIDES HPD, APEH, ALDH7A1 KDM4E 664/4885ALDH1A1 36/4885MAPT 4149/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.