SCHEMBL5485178

SCHEMBL5485178

COC(=O)C(Cl)c1ccc(Br)c(C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
RAB9A P51151 3/20 0.42
NPC1 O15118 2/20 0.42
SLC6A3 Q01959 2/20 0.42
MAPT P10636 1/20 0.42
CHRNA1 P02708 1/20 0.42
CHRNG P07510 1/20 0.42
CHRNB1 P11230 1/20 0.42
CHRNB2 P17787 1/20 0.42
SLC6A2 P23975 1/20 0.42
CHRNB4 P30926 1/20 0.42
SLC6A4 P31645 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA4 P43681 1/20 0.42
CHRND Q07001 1/20 0.42
PKM P14618 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
KMT2A Q03164 4/20 0.38
MT-CO2 P00403 1/20 0.38
MEN1 O00255 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL850725 0.83 ALDH1A1 (0.45) ALDH1A1RAB9ANPC1SLC6A3MAPT
SCHEMBL7098148 0.82 MT-CO2 (0.55) ALDH1A1RAB9ANPC1SLC6A3MAPT
SCHEMBL25980311 0.78 ALDH1A1 (0.41) ALDH1A1RAB9ANPC1SLC6A3MAPT
SCHEMBL803625 0.77 TAS1R3 (0.46) ALDH1A1KMT2AMEN1CYP2C19LMNA
SCHEMBL8926621 0.76 TSHR (0.48) ALDH1A1RAB9ANPC1MAPTSMN1; SMN2
SCHEMBL4779827 0.75 L3MBTL1 (0.49) ALDH1A1SMN1; SMN2KMT2AMT-CO2MEN1
SCHEMBL5487986 0.75 SLC6A3 (0.57) ALDH1A1SLC6A3SLC6A2SLC6A4SMN1; SMN2
SCHEMBL11458699 0.74 CYP1A2 (0.42) SLC6A3MAPTCYP1A2CYP2C9LMNA
SCHEMBL187559 0.73 CYP2C19 (0.52) ALDH1A1SMN1; SMN2KMT2ACYP1A2CYP3A4
SCHEMBL11469391 0.72 SLC6A3 (0.50) SLC6A3KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7256158-B2 2,4,5,-trisubstituted phenylketo-enols for use as pesticides and herbicides BAYER AG (DE) 2007-08-14 US disclosed
US-6933261-B2 2,4,5-Trisubstituted phenylketoenols BAYER AKTIENGESELLSCHAFT (DE) 2005-08-23 US disclosed
US-20050038021-A1 2,4,5,-trisubstituted phenylketo-enols for use as pesticides and herbicides BAYER AG (DE) 2005-02-17 US disclosed
US-20030171219-A1 2,4,5-trisubstituted phenylketo-enols for use as pesticides and herbicides LIEB FOLKER (DE) 2003-09-11 US disclosed
US-6511942-B1 Animal husbandry, veterinary medicine BAYER AKTIENGESELLSCHAFT (DE) 2003-01-28 US disclosed
US-6110872-A 3-(2,4,5-TRISUBSTITUTED PHENYL), 4-HYDROXY,5,5-(CYCLOALKYL OR HETEROCYCLOALKYL)PYRROLIN-2-ONE AND DERIVATIVES; METHOD OF MAKING BY INTRAMOLECULAR CONDENSATION OF SPECIFIED COMPOUND BAYER AKTIENGESELLSCHAFT (DE) 2000-08-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050038021-A1 2,4,5,-trisubstituted phenylketo-enols for use as pesticides and herbicides DDT, CYP4X1, PDHX ALDH1A1 1592/4885RAB9A 4145/4885NPC1 4575/4885
US-20030171219-A1 2,4,5-trisubstituted phenylketo-enols for use as pesticides and herbicides DDT, CYP4X1, HPD ALDH1A1 855/4885RAB9A 4214/4885NPC1 4175/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.