SCHEMBL5493334

SCHEMBL5493334

COC(=O)C1C(=O)CCC1(C)C

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TSHR P16473 2/20 0.40
ALDH1A1 P00352 7/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
ALOX12 P18054 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
HIF1A Q16665 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4135825 0.89 ALDH1A1 (0.40) GAAMAPTNPSR1TSHRALDH1A1
SCHEMBL2264463 0.80 ALDH1A1 (0.40) GAAMAPTTSHRALDH1A1ALOX12
SCHEMBL2567271 0.78 TSHR (0.38) GAAMAPTNPSR1TSHRALDH1A1
SCHEMBL27792315 0.78 APLNR (0.33) HTTKMT2AMEN1
SCHEMBL5500597 0.77 DNTT (0.35) GAAMAPTNPSR1TSHRALDH1A1
SCHEMBL9851192 0.74 GAA (0.47) GAAMAPTNPSR1TSHRALDH1A1
SCHEMBL30585217 0.73 PTPN2 (0.43) GAAMAPTNPSR1TSHRALDH1A1
SCHEMBL30585215 0.73 PTPN2 (0.43) GAAMAPTNPSR1TSHRALDH1A1
SCHEMBL9609154 0.73 PTPN2 (0.43) GAAMAPTNPSR1TSHRALDH1A1
SCHEMBL8514874 0.73 PTPN2 (0.43) GAAMAPTNPSR1TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4142732-B1 METHODS OF USE FOR PYRIMIDINES AS FERROPORTIN INHIBITORS GLOBAL BLOOD THERAPEUTICS INC (US) 2026-04-22 EP disclosed
US-20250109122-A1 CYCLOALKYL PYRIMIDINES AS FERROPORTIN INHIBITORS GLOBAL BLOOD THERAPEUTICS INC (US) 2025-04-03 US disclosed
US-12202817-B2 Cycloalkyl pyrimidines as ferroportin inhibitors GLOBAL BLOOD THERAPEUTICS, INC. (US) 2025-01-21 US disclosed
US-12037322-B2 AHR agonists ELI LILLY AND COMPANY (US) 2024-07-16 US disclosed
CN-118215654-A AHR agonists 伊莱利利公司 2024-06-18 CN disclosed
US-20240140932-A1 CYCLOALKYL PYRIMIDINES AS FERROPORTIN INHIBITORS GLOBAL BLOOD THERAPEUTICS INC (US) 2024-05-02 US disclosed
US-11834421-B2 Saturated-ring-fused dihydropyrimidinone or dihydrotriazinone compounds and pharmaceutical use thereof JAPAN TOBACCO INC. (JP) 2023-12-05 US disclosed
US-11834421-B2 Saturated-ring-fused dihydropyrimidinone or dihydrotriazinone compounds and pharmaceutical use thereof JAPAN TOBACCO INC. (JP) 2023-12-05 US disclosed
CN-111741948-B Saturated ring-fused dihydropyrimidinone or dihydrotriazinone compounds and pharmaceutical use thereof 日本烟草产业株式会社 2023-11-10 CN disclosed
EP-3760619-B1 SATURATED RING-CONDENSED DIHYDROPYRIMIDINONE OR DIHYDROTRIAZINONE COMPOUND, AND PHARMACEUTICAL USE THEREOF JAPAN TOBACCO INC (JP) 2023-10-25 EP disclosed
US-20170197941-A1 CYCLOHEXEN-1-YL-PYRIDIN-2-YL-1H-PYRAZOLE-4-CARBOXYLIC ACID DERIVATIVES AND THE USE THEREOF AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS NOVARTIS AG (CH) 2017-07-13 US disclosed
EP-1790644-A1 Substituted benzopyrans as selective estrogen receptor-beta agonists ELI LILLY AND COMPANY (US) 2007-05-30 EP disclosed
EP-1448544-B1 SUBSTITUTED BENZOPYRANS AS SELECTIVE ESTROGEN RECEPTOR-BETA AGONISTS LILLY CO ELI (US) 2007-05-16 EP disclosed
US-7217734-B2 Substituted benzopyrans as selective estrogen receptor-beta agonists ELI LILLY AND COMPANY (US) 2007-05-15 US disclosed
CN-1312147-C Substituted benzopyrans as selective estrogen receptor-beta agonists LILLY CO ELI (US) 2007-04-25 CN disclosed
CN-1589268-A Substituted benzopyrans as selective estrogen receptor-beta agonists LILLY CO ELI (US) 2005-03-02 CN disclosed
US-20040249167-A1 Substituted benzopyrans as selective estrogen receptor-beta agonists ELI LILLY AND COMPANY 2004-12-09 US disclosed
EP-1448544-A1 SUBSTITUTED BENZOPYRANS AS SELECTIVE ESTROGEN RECEPTOR-BETA AGONISTS ELI LILLY AND COMPANY (US) 2004-08-25 EP disclosed
US-6630508-B1 For treating prostate cancer ELI LILLY AND COMPANY 2003-10-07 US disclosed
WO-2003044006-A1 SUBSTITUTED BENZOPYRANS AS SELECTIVE ESTROGEN RECEPTOR-BETA AGONISTS ELI LILLY AND COMPANY (US) 2003-05-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11834421-B2 Saturated-ring-fused dihydropyrimidinone or dihydrotriazinone compounds and pharmaceutical use thereof RORC, RORB, RORA GAA 2685/4885MAPT 1809/4885NPSR1 253/4885
US-12202817-B2 Cycloalkyl pyrimidines as ferroportin inhibitors HAMP, SLC40A1, FANCI GAA 1395/4885MAPT 4441/4885NPSR1 3095/4885
US-20170197941-A1 CYCLOHEXEN-1-YL-PYRIDIN-2-YL-1H-PYRAZOLE-4-CARBOXYLIC ACID DERIVATIVES AND THE USE THEREOF AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS GUCY1A1, GUCY1A2, GUCY1B2 GAA 805/4885MAPT 3714/4885NPSR1 1983/4885
US-20040249167-A1 Substituted benzopyrans as selective estrogen receptor-beta agonists GPER1, ESR1, ESR2 GAA 2476/4885MAPT 3336/4885NPSR1 44/4885
US-12037322-B2 AHR agonists AHR, ARNT, RORC GAA 3710/4885MAPT 3658/4885NPSR1 336/4885
US-20250109122-A1 CYCLOALKYL PYRIMIDINES AS FERROPORTIN INHIBITORS HAMP, SLC40A1, FANCI GAA 1395/4885MAPT 4441/4885NPSR1 3095/4885
US-20240140932-A1 CYCLOALKYL PYRIMIDINES AS FERROPORTIN INHIBITORS HAMP, SLC40A1, FANCI GAA 1395/4885MAPT 4441/4885NPSR1 3095/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.