SCHEMBL5500897

SCHEMBL5500897

NC(=O)N(CCNc1ccc(OC(F)(F)F)cc1)C(=O)[CH]CSCc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.42
CTSS P25774 2/20 0.40
CTSL P07711 1/20 0.40
CTSK P43235 1/20 0.40
FPR2 P25090 1/20 0.39
MAPT P10636 2/20 0.38
PLA2G1B P04054 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ATG4B Q9Y4P1 1/20 0.38
HDAC1 Q13547 2/20 0.37
HTT P42858 2/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
RAB9A P51151 1/20 0.37
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.36
GRIN2B Q13224 1/20 0.36
ACHE P22303 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5398970 0.82 CTSS (0.41) EPHX1CTSSFPR2MAPTPLA2G1B
SCHEMBL3024779 0.77 CTSS (0.49) EPHX1CTSSCTSLCTSKFPR2
SCHEMBL6685716 0.75 KDM4E (0.47) EPHX1CTSSCTSLCTSKPOLB
SCHEMBL5500899 0.71 EPHX1 (0.52) EPHX1CTSSCTSLCTSKFPR2
SCHEMBL24327967 0.69 FPR2 (0.52) FPR2MAPTPLA2G1BSMN1; SMN2ATG4B
SCHEMBL6691065 0.69 RAB9A (0.45) CTSSCTSKMAPTSMN1; SMN2KMT2A
SCHEMBL3024781 0.68 CTSS (0.67) CTSSCTSLCTSKACE
SCHEMBL6689992 0.67 CFD (0.41) EPHX1POLBEPHX2
SCHEMBL9422891 0.66 ACHE (0.61) MAPTPLA2G1BSMN1; SMN2ATG4BHTT
SCHEMBL6688710 0.65 POLB (0.43) EPHX1MAPTHDAC1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658267-A4 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2007-08-01 EP disclosed
EP-1658267-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2006-05-24 EP disclosed
WO-2005034848-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2005-04-21 WO disclosed