SCHEMBL5508962

SCHEMBL5508962

COC(=O)C1CCN(C(=O)O)C1c1cc(NC(C)=O)ccc1O

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.41
MTNR1A P48039 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HTR1A P08908 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
HTR1F P30939 1/20 0.38
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
RORC P51449 1/20 0.36
KDM4E B2RXH2 1/20 0.36
HTT P42858 1/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5508963 0.81 DRD2 (0.42) TSHRSLC6A2SLC6A4SLC6A3
SCHEMBL8262944 0.68 DRD2 (0.42) TSHRSLC6A2SLC6A4SLC6A3
SCHEMBL5508811 0.67 SLC6A4 (0.39) TSHRSLC6A2SLC6A4SLC6A3
SCHEMBL5531271 0.67 SLC6A4 (0.38) TSHRSLC6A2SLC6A4SLC6A3
SCHEMBL2944250 0.67 NPC1 (0.52)
SCHEMBL4110657 0.66 F7 (0.39) TSHRSLC6A2SLC6A4SLC6A3
SCHEMBL5508290 0.64 LMNA (0.43) TSHRHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL5508296 0.64 LMNA (0.43) TSHRHTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL20899353 0.63 AR (0.39) TSHRSMN1; SMN2SLC6A2SLC6A4SLC6A3
SCHEMBL4591071 0.63 NPC1 (0.53) SMN1; SMN2HTR1AKDM4ESLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856096-A2 PHENYLGLYCINAMIDE DERIVATIVES USEFUL AS ANTICOAGULANTS Bristol-Myers Squibb Company (US) 2007-11-21 EP disclosed
WO-2006076246-A2 PHENYLGLYCINAMIDE DERIVATIVES USEFUL AS ANTICOAGULANTS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-20 WO disclosed