SCHEMBL5524698

SCHEMBL5524698

CCC(=O)Nc1cccc(C(N)=O)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.71
MEN1 O00255 5/20 0.71
L3MBTL1 Q9Y468 1/20 0.69
PARP1 P09874 5/20 0.67
PARP10 Q53GL7 4/20 0.67
RAB9A P51151 2/20 0.63
POLB P06746 1/20 0.63
NR4A1 P22736 1/20 0.63
ALDH1A1 P00352 3/20 0.62
MAPK1 P28482 1/20 0.62
GAA P10253 1/20 0.61
LMNA P02545 3/20 0.58
SMN1; SMN2 Q16637 3/20 0.58
CYP1A2 P05177 1/20 0.58
MAPT P10636 1/20 0.58
CYP2C19 P33261 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
SMYD3 Q9H7B4 1/20 0.58
PARP14 Q460N5 1/20 0.57
NPC1 O15118 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30716404 1.00 KMT2A (0.71) KMT2AMEN1L3MBTL1PARP1PARP10
SCHEMBL3362788 0.87 MEN1 (0.77) KMT2AMEN1L3MBTL1PARP1PARP10
SCHEMBL18671651 0.86 KMT2A (0.87) KMT2AMEN1L3MBTL1PARP1PARP10
SCHEMBL5820518 0.86 L3MBTL1 (0.73) KMT2AMEN1L3MBTL1RAB9APOLB
SCHEMBL11545396 0.85 PARP1 (0.74) KMT2AMEN1L3MBTL1PARP1PARP10
SCHEMBL10964661 0.85 L3MBTL1 (0.77) KMT2AMEN1L3MBTL1RAB9APOLB
Benzamide SCHEMBL27225883 0.85 ALDH1A1 (0.68) KMT2AMEN1L3MBTL1PARP1RAB9A
SCHEMBL11803436 0.85 L3MBTL1 (0.71) KMT2AMEN1L3MBTL1RAB9APOLB
SCHEMBL3646401 0.85 MEN1 (0.73) KMT2AMEN1L3MBTL1PARP1PARP10
SCHEMBL10970617 0.84 RAB9A (0.85) KMT2AMEN1L3MBTL1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230346946-A1 Nanostructured Gels Capable of Controlled Release of Encapsulated Agents THE BRIGHAM AND WOMEN'S HOSPITAL, INC. 2023-11-02 US disclosed
US-11672864-B2 Nanostructured gels capable of controlled release of encapsulated agents THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2023-06-13 US disclosed
US-10675351-B2 Nanostructured gels capable of controlled release of encapsulated agents THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2020-06-09 US disclosed
US-9974859-B2 Nanostructured gels capable of controlled release of entrapped agents THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2018-05-22 US disclosed
US-9974859-B2 Nanostructured gels capable of controlled release of entrapped agents THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2018-05-22 US disclosed
US-20170000888-A1 NANOSTRUCTURED GELS CAPABLE OF CONTROLLED RELEASE OF ENTRAPPED AGENTS THE BRIGHAM AND WOMEN'S HOSPITAL, INC. 2017-01-05 US disclosed
US-8288540-B2 2-heteroarylamino-pyrimidine derivatives as kinase inhibitors IRM LLC (BM) 2012-10-16 US disclosed
US-20110053952-A1 2-HETEROARYLAMINO-PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS IRM LLC (BM) 2011-03-03 US disclosed
US-20090264649-A1 DIARYLAMINE-CONTAINING COMPOUNDS AND COMPOSITIONS, AND THEIR USE AS MODULATORS OF C-KIT RECEPTORS IRM LLC (BM) 2009-10-22 US disclosed
US-7592349-B2 Diarylamine-containing compounds and compositions, and their use as modulators of c-kit receptors IRM LLC (BM) 2009-09-22 US disclosed
US-20080167308-A1 DIARYLAMINE-CONTAINING COMPOUNDS AND COMPOSITIONS, AND THEIR USE AS MODULATORS OF C-KIT RECEPTORS IRM LLC, A DELAWARE LIMITED LIABILITY COMAPNY (BM) 2008-07-10 US disclosed
US-20080139559-A1 DIARYLAMINE-CONTAINING COMPOUNDS AND COMPOSITIONS, AND THEIR USE AS MODULATORS OF C-KIT RECEPTORS IRM LLC, A DELAWARE LIMITED LIABILITY COMAPNY (BM) 2008-06-12 US disclosed
US-20080139597-A1 DIARYLAMINE-CONTAINING COMPOUNDS AND COMPOSITIONS, AND THEIR USE AS MODULATORS OF C-KIT RECEPTORS IRM LLC, A DELAWARE LIMITED LIABILITY COMAPNY (BM) 2008-06-12 US disclosed
US-20070149538-A1 Diarylamine-Containing Compounds and Compositions, and their use as Modulators of C-Kit Receptors IRM LLC (BM) 2007-06-28 US disclosed
US-20070010671-A1 Novel quinazoline derivatives and methods of treatment related to the use thereof ARENA PHARMACEUTICALS, INC. 2007-01-11 US disclosed
US-5719151-A PHTHALAZINEDIONE COMPOUND; POLYMERASE INHIBITOR SHALL SYDNEY (GB) 1998-02-17 US disclosed
US-5633282-A ENZYME INHIBITORS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1997-05-27 US disclosed
EP-0531370-B1 INHIBITION OF VIRAL INFECTION BRITISH TECH GROUP (GB) 1996-09-18 EP disclosed
EP-0531370-A1 INHIBITION OF VIRAL INFECTION. COLLINS MARY KATHARINE LEVINGE (GB) 1993-03-17 EP disclosed
WO-1991018591-A1 INHIBITION OF VIRAL INFECTION COLLINS MARY KATHARINE LEVINGE (GB) 1991-12-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230346946-A1 Nanostructured Gels Capable of Controlled Release of Encapsulated Agents MMP2, CEL, LIPA KMT2A 3895/4885MEN1 3515/4885L3MBTL1 4251/4885
US-20090264649-A1 DIARYLAMINE-CONTAINING COMPOUNDS AND COMPOSITIONS, AND THEIR USE AS MODULATORS OF C-KIT RECEPTORS KIT, PRKCH, PRKCE KMT2A 646/4885MEN1 2421/4885L3MBTL1 4630/4885
US-20070010671-A1 Novel quinazoline derivatives and methods of treatment related to the use thereof MCHR1, GPR119, MCHR2 KMT2A 792/4885MEN1 647/4885L3MBTL1 3309/4885
US-20080139597-A1 DIARYLAMINE-CONTAINING COMPOUNDS AND COMPOSITIONS, AND THEIR USE AS MODULATORS OF C-KIT RECEPTORS KIT, PRKCH, PRKCE KMT2A 646/4885MEN1 2421/4885L3MBTL1 4630/4885
US-20110053952-A1 2-HETEROARYLAMINO-PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS FYN, LCK, ERBB2 KMT2A 1233/4885MEN1 4779/4885L3MBTL1 3713/4885
US-20170000888-A1 NANOSTRUCTURED GELS CAPABLE OF CONTROLLED RELEASE OF ENTRAPPED AGENTS MMP2, MMP1, GUSB KMT2A 4034/4885MEN1 3859/4885L3MBTL1 4245/4885
US-20070149538-A1 Diarylamine-Containing Compounds and Compositions, and their use as Modulators of C-Kit Receptors KIT, PRKCH, PRKCE KMT2A 646/4885MEN1 2421/4885L3MBTL1 4630/4885
US-10675351-B2 Nanostructured gels capable of controlled release of encapsulated agents MMP2, CEL, LIPA KMT2A 3895/4885MEN1 3515/4885L3MBTL1 4251/4885
US-20080167308-A1 DIARYLAMINE-CONTAINING COMPOUNDS AND COMPOSITIONS, AND THEIR USE AS MODULATORS OF C-KIT RECEPTORS KIT, PRKCH, PRKCE KMT2A 646/4885MEN1 2421/4885L3MBTL1 4630/4885
US-11672864-B2 Nanostructured gels capable of controlled release of encapsulated agents MMP2, CEL, LIPA KMT2A 3895/4885MEN1 3515/4885L3MBTL1 4251/4885
US-20080139559-A1 DIARYLAMINE-CONTAINING COMPOUNDS AND COMPOSITIONS, AND THEIR USE AS MODULATORS OF C-KIT RECEPTORS KIT, PRKCH, PRKCE KMT2A 646/4885MEN1 2421/4885L3MBTL1 4630/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.