SCHEMBL5533178

SCHEMBL5533178

CC1=C(C(=O)O)C(c2cc(Cl)ccc2Cl)(C(C)(C)C)C(C(=O)O)=C(C)N1C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.39
ALDH1A1 P00352 3/20 0.36
TP53 P04637 1/20 0.36
NOTUM Q6P988 3/20 0.36
HTT P42858 1/20 0.34
MYC P01106 2/20 0.33
NR4A1 P22736 1/20 0.33
TSHR P16473 1/20 0.33
CASP1 P29466 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
LMNA P02545 2/20 0.32
NPC1 O15118 1/20 0.32
PKM P14618 1/20 0.32
PDK1 Q15118 1/20 0.31
PDK2 Q15119 1/20 0.31
PDK3 Q15120 1/20 0.31
PDK4 Q16654 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CTSB P07858 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4757311 0.81 TSHR (0.37) ALDH1A1NOTUMTSHRLMNAPDK1
SCHEMBL4814956 0.75 ALDH1A1 (0.32) ALDH1A1MYCNR4A1SMN1; SMN2PKM
SCHEMBL4826843 0.69 HCAR3 (0.39) HCAR2ALDH1A1HTTMYCNR4A1
SCHEMBL4757320 0.67 HCAR2 (0.39) HCAR2ALDH1A1TP53NOTUMHTT
SCHEMBL4757323 0.62 SMN1; SMN2 (0.40) HCAR2ALDH1A1TP53NOTUMHTT
SCHEMBL4758286 0.59 TSHR (0.36) HCAR2ALDH1A1TP53NOTUMHTT
SCHEMBL4758043 0.58 CRHBP (0.40) ALDH1A1TP53NOTUMHTTSMN1; SMN2
SCHEMBL224469 0.56 ALDH1A1 (1.00) ALDH1A1TP53NOTUMMYCNR4A1
Acetic Acid SCHEMBL27374496 0.56 TP53 (0.67) ALDH1A1TP53HTTTSHRCASP1
SCHEMBL6584266 0.55 ALDH1A1 (0.95) ALDH1A1TP53NOTUMMYCNR4A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1858325-A2 COMPOUNDS FOR INHIBITING BETA-AMYLOID PRODUCTION AND METHODS OF IDENTIFYING THE COMPOUNDS Roskamp Research LLC (US) 2007-11-28 EP disclosed
WO-2006074419-A2 COMPOUNDS FOR INHIBITING BETA-AMYLOID PRODUCTION AND METHODS OF IDENTIFYING THE COMPOUNDS ROSKAMP RESEARCH LLC (US) 2006-07-13 WO disclosed