SCHEMBL4757320

SCHEMBL4757320

CCN1C(C)=C(C(=O)O)C(CC)(c2cc(Cl)ccc2Cl)C(C(=O)O)=C1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.39
ALDH1A1 P00352 3/20 0.38
LMNA P02545 2/20 0.38
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.36
NOTUM Q6P988 2/20 0.36
HTT P42858 2/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.34
MYC P01106 2/20 0.33
TSHR P16473 2/20 0.33
CASP1 P29466 2/20 0.33
NR4A1 P22736 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MARS1 P56192 1/20 0.33
KCNK2 O95069 1/20 0.33
GAA P10253 2/20 0.33
GFER P55789 1/20 0.33
THRB P10828 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4758286 0.90 TSHR (0.36) HCAR2ALDH1A1LMNAMAPTTP53
SCHEMBL4757355 0.84 PYGM (0.39) ALDH1A1LMNANOTUMHTTGAA
SCHEMBL4757333 0.81 OPRM1 (0.36) ALDH1A1NOTUMTSHRSMN1; SMN2GAA
SCHEMBL4758575 0.81 OPRM1 (0.39) NOTUMTSHR
SCHEMBL4758254 0.80 HCAR3 (0.39) HCAR2ALDH1A1LMNAMAPTNOTUM
SCHEMBL4758577 0.80 TSHR (0.36) ALDH1A1LMNAMAPTTP53NOTUM
SCHEMBL4758583 0.79 PYGL (0.38) ALDH1A1LMNAMAPTNOTUMTSHR
SCHEMBL4757340 0.79 NOTUM (0.34) NOTUM
SCHEMBL5533759 0.78 KDM4E (0.39) ALDH1A1LMNAMAPTHTTTSHR
SCHEMBL5452071 0.76 ABCC1 (0.43) HCAR2ALDH1A1LMNAMAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008006070-A2 COMPOUNDS AND COMBINATIONS THEREOF FOR INHIBITING BETA-AMYLOID PRODUCTION AND METHODS OF USE THEREOF ROSKAMP RESEARCH LLC (US) 2008-01-10 WO disclosed