SCHEMBL5535948

SCHEMBL5535948

Cc1nc(-c2ccc(N3CC(CN4CCN(OC(=O)Nc5ccc(Cl)c(Cl)c5)CC4)OC3=O)cc2)no1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 3/20 0.40
KCNH2 Q12809 3/20 0.40
SIGMAR1 Q99720 10/20 0.40
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
LMNA P02545 1/20 0.40
DGAT1 O75907 1/20 0.38
THRB P10828 1/20 0.38
MAPK14 Q16539 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5533939 0.89 THRB (0.44) SIGMAR1ITGB3ITGA2BLMNATHRB
SCHEMBL5535143 0.86 ITGB3 (0.37) SIGMAR1ITGB3ITGA2BLMNADGAT1
SCHEMBL5530623 0.84 SIGMAR1 (0.45) SIGMAR1ITGB3ITGA2BDGAT1THRB
SCHEMBL7387348 0.80 MAPT (0.49) CCR2KCNH2SIGMAR1LMNADGAT1
SCHEMBL5530617 0.78 SIGMAR1 (0.45) SIGMAR1ITGB3ITGA2BDGAT1THRB
SCHEMBL7389109 0.77 THRB (0.51) SIGMAR1LMNATHRB
SCHEMBL7388632 0.76 THRB (0.46) SIGMAR1ITGB3ITGA2BLMNATHRB
SCHEMBL7389681 0.76 THRB (0.46) SIGMAR1LMNATHRB
SCHEMBL7386854 0.76 DGAT1 (0.42) SIGMAR1ITGB3ITGA2BLMNADGAT1
SCHEMBL7388647 0.76 MAPT (0.48) SIGMAR1LMNATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1416931-B1 INHIBITORS OF POLYQ-AGGREGATION MAX PLANCK GESELLSCHAFT (DE) 2007-06-13 EP claimed