SCHEMBL5535143

SCHEMBL5535143

Cc1nc(-c2ccc(N3CC(CN4CCN(OC(=O)Nc5ccc(F)c([N+](=O)[O-])c5)CC4)OC3=O)cc2)no1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
RAC1 P63000 1/20 0.37
SIGMAR1 Q99720 9/20 0.36
PIK3CD O00329 1/20 0.36
AKT1 P31749 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
MAPK14 Q16539 2/20 0.36
POLB P06746 2/20 0.36
MAPT P10636 2/20 0.36
TP53 P04637 1/20 0.36
ALDH1A1 P00352 2/20 0.35
MAOA P21397 2/20 0.35
DGAT1 O75907 1/20 0.35
GAA P10253 1/20 0.35
LMNA P02545 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PTGS1 P23219 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5535948 0.86 CCR2 (0.40) ITGB3ITGA2BSIGMAR1MAPK14DGAT1
SCHEMBL5533939 0.85 THRB (0.44) ITGB3ITGA2BSIGMAR1MAPK14MAPT
SCHEMBL5530623 0.80 SIGMAR1 (0.45) ITGB3ITGA2BSIGMAR1DGAT1
SCHEMBL7389426 0.77 THRB (0.45) POLBMAPTALDH1A1LMNAMEN1
SCHEMBL7380624 0.76 PKM (0.44) SIGMAR1PIK3CAPOLBMAPTALDH1A1
SCHEMBL7592402 0.76 MAPT (0.46) SIGMAR1POLBMAPTTP53MAOA
SCHEMBL7387348 0.75 MAPT (0.49) SIGMAR1POLBMAPTDGAT1LMNA
SCHEMBL7386967 0.75 MAPT (0.44) SIGMAR1POLBMAPTTP53DGAT1
SCHEMBL5530617 0.74 SIGMAR1 (0.45) ITGB3ITGA2BSIGMAR1DGAT1
SCHEMBL7387692 0.73 THRB (0.42) SIGMAR1MAPTALDH1A1GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1416931-B1 INHIBITORS OF POLYQ-AGGREGATION MAX PLANCK GESELLSCHAFT (DE) 2007-06-13 EP claimed