SCHEMBL5558540

SCHEMBL5558540

NCc1ccc(-c2ccc(Cl)c(Cl)c2)cc1

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.62
AHR P35869 3/20 0.61
HRH3 Q9Y5N1 1/20 0.61
CYP1B1 Q16678 1/20 0.52
PNMT P11086 3/20 0.52
MAOB P27338 2/20 0.47
IDO1 P14902 3/20 0.45
S1PR1 P21453 1/20 0.45
S1PR5 Q9H228 1/20 0.45
CSNK2A1 P68400 2/20 0.44
PTPN5 P54829 1/20 0.43
SIGMAR1 Q99720 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL29385902 0.82 TAAR1 (0.68) TAAR1AHRPNMTMAOBSIGMAR1
SCHEMBL29349576 0.81 PNMT (0.67) TAAR1PNMTIDO1CSNK2A1SIGMAR1
SCHEMBL112200 0.81 PNMT (0.67) TAAR1PNMTIDO1CSNK2A1SIGMAR1
SCHEMBL11071591 0.80 AHR (0.64) TAAR1AHRCYP1B1PNMTIDO1
Ammonia Solution, Strong SCHEMBL9178453 0.79 PNMT (0.64) TAAR1PNMTIDO1CSNK2A1SIGMAR1
Hydrochloric Acid SCHEMBL3127848 0.79 PNMT (0.64) TAAR1PNMTIDO1CSNK2A1SIGMAR1
SCHEMBL27717640 0.79 TAAR1 (0.53) TAAR1AHRHRH3PNMTMAOB
SCHEMBL8024771 0.78 AHR (0.61) TAAR1AHRCYP1B1PNMTIDO1
SCHEMBL12603805 0.78 AHR (0.61) TAAR1AHRCYP1B1PNMTIDO1
SCHEMBL2274647 0.78 HRH3 (1.00) TAAR1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8470859-B2 Iminopyridine derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-06-25 US disclosed
US-8470859-B2 Iminopyridine derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-06-25 US disclosed
US-20100016315-A1 Iminopyridine Derivative and Use Thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-01-21 US disclosed
US-20100016315-A1 Iminopyridine Derivative and Use Thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-01-21 US disclosed
US-20070197577-A1 Inhibitors of anthrax lethal factor CENGENT THERAPEUTICS (US) 2007-08-23 US disclosed
WO-2005027856-A2 INHIBITORS OF ANTHRAX LETHAL FACTOR CENGENT THERAPEUTICS (US) 2005-03-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100016315-A1 Iminopyridine Derivative and Use Thereof ADRA1D, ADRB1, ADRB2 TAAR1 122/4885AHR 980/4885HRH3 500/4885
US-20070197577-A1 Inhibitors of anthrax lethal factor APAF1, ANTXR2, LITAF TAAR1 4731/4885AHR 2502/4885HRH3 2936/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.