SCHEMBL5585773

SCHEMBL5585773

CC(=O)OC1(NC(=O)c2ccccc2)CCCCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.48
ADRB2 P07550 1/20 0.47
CTSL P07711 4/20 0.46
ALDH1A1 P00352 3/20 0.43
HTT P42858 2/20 0.43
KDM4E B2RXH2 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
APAF1 O14727 1/20 0.43
TDP2 O95551 1/20 0.43
NSD2 O96028 1/20 0.43
ABL1 P00519 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HSP90AB1 P08238 1/20 0.43
MAPT P10636 1/20 0.43
CASP3 P42574 1/20 0.43
GALK1 P51570 1/20 0.43
BLM P54132 1/20 0.43
PPP1CA P62136 1/20 0.43
RIN1 Q13671 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3645705 0.95 ALDH1A1 (0.44) CTSKADRB2CTSLALDH1A1HTT
SCHEMBL5586066 0.85 ALDH1A1 (0.45) CTSKCTSLALDH1A1HTTKDM4E
SCHEMBL9009913 0.79 RAB9A (0.45) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL27797797 0.77 CTSL (0.42) CTSKADRB2CTSLALDH1A1HTT
SCHEMBL9009877 0.77 ALDH1A1 (0.51) ALDH1A1HTTKDM4EMEN1KMT2A
SCHEMBL27743186 0.77 KMT2A (0.41) CTSLALDH1A1HTTKDM4EMEN1
SCHEMBL27712467 0.76 IDO1 (0.42) CTSKCTSLMEN1KMT2AMAPT
SCHEMBL10590807 0.76 CTSK (0.54) CTSKADRB2CTSLALDH1A1HTT
SCHEMBL11609600 0.76 ALDH1A1 (0.54) CTSKADRB2CTSLALDH1A1HTT
SCHEMBL9009859 0.75 HTT (0.37) ALDH1A1HTTMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976932-A Fused quinoline derivative and use thereof TAKEDA PHARMACEUTICAL (JP) 2007-06-06 CN disclosed
EP-1740584-A1 FUSED QUINOLINE DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-01-10 EP disclosed
WO-2005105802-A1 FUSED QUINOLINE DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-10 WO disclosed