SCHEMBL565913

SCHEMBL565913

COc1ccc2c(c1)CCN2

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.53
DRD4 P21917 1/20 0.53
PDE3B Q13370 1/20 0.51
PDE3A Q14432 1/20 0.51
HRH3 Q9Y5N1 1/20 0.49
HTR2C P28335 2/20 0.49
HTR2A P28223 1/20 0.46
HTR2B P41595 1/20 0.46
BCL2 P10415 1/20 0.46
TNIK Q9UKE5 1/20 0.44
ALDH1A1 P00352 1/20 0.43
DRD1 P21728 1/20 0.43
DRD5 P21918 1/20 0.43
DRD3 P35462 1/20 0.43
SNCA P37840 1/20 0.43
ACHE P22303 1/20 0.43
APP P05067 1/20 0.43
KCNH2 Q12809 1/20 0.42
RYR2 Q92736 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2208190 0.98 DRD2 (0.52) DRD2DRD4PDE3BPDE3AHRH3
Hydrochloric Acid SCHEMBL2208192 0.98 DRD2 (0.52) DRD2DRD4PDE3BPDE3AHRH3
SCHEMBL665048 0.89 CA12 (0.53) DRD2DRD4PDE3BPDE3AHRH3
Hydrochloric Acid SCHEMBL8021718 0.87 KDM4E (0.53) DRD2DRD4PDE3BPDE3AHRH3
SCHEMBL2778234 0.87 HRH3 (0.48) DRD2DRD4PDE3BPDE3AHRH3
Hydrochloric Acid SCHEMBL3526192 0.86 KDM4E (0.48) DRD2DRD4PDE3BPDE3AHRH3
SCHEMBL30025932 0.85 HTR2C (0.50) DRD2PDE3BPDE3AHRH3HTR2C
SCHEMBL550150 0.85 HTR2C (0.50) DRD2PDE3BPDE3AHRH3HTR2C
SCHEMBL20956992 0.82 TNIK (0.56) DRD2DRD4HTR2CHTR2BTNIK
SCHEMBL12079387 0.82 PDE3B (0.61) PDE3BPDE3AHTR2CBCL2TNIK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 240 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117229275-B Novel 2-acetamido thiazole compound and preparation method and application thereof 北京中医药大学 2024-06-18 CN claimed
CN-115626889-B Organic chemical conversion method for oxidative dehydrogenation of nitrogen-containing heterocyclic compound 南京工业大学 2024-04-30 CN claimed
CN-115353478-A Preparation method of indole compound 南京工业大学 2022-11-18 CN claimed
CN-115160824-A Method for preparing multicolor dye from single polymer 四川大学 2022-10-11 CN claimed
US-20190127345-A1 NEGATIVE PHOTOCHROMIC MATERIALS WITH TUNABLE PROPERTIES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-05-02 US claimed
WO-2017189700-A1 NEGATIVE PHOTOCHROMIC MATERIALS WITH TUNABLE PROPERTIES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-11-02 WO claimed
JP-9278752-A None JP disclosed
EP-4142732-B1 METHODS OF USE FOR PYRIMIDINES AS FERROPORTIN INHIBITORS GLOBAL BLOOD THERAPEUTICS INC (US) 2026-04-22 EP disclosed
US-12599584-B2 Indoline derivatives, compositions comprising them and uses thereof YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. (IL) 2026-04-14 US disclosed
EP-4692071-A1 PHOTOCHROMIC COMPOUND, NAPHTHOL DERIVATIVE, CURABLE COMPOSITION, OPTICAL ARTICLE, LENS, AND EYEGLASS TOKUYAMA CORPORATION (JP) 2026-02-11 EP disclosed
US-20250122152-A1 KAT6 Inhibitors BEIGENE SWITZERLAND GMBH (CH) 2025-04-17 US disclosed
US-20250109122-A1 CYCLOALKYL PYRIMIDINES AS FERROPORTIN INHIBITORS GLOBAL BLOOD THERAPEUTICS INC (US) 2025-04-03 US disclosed
WO-2025068943-A1 KAT6 INHIBITORS BEIGENE SWITZERLAND GMBH (CH) 2025-04-03 WO disclosed
EP-0159376-A1 1-(Aminoalkylphenyl and Aminoalkylbenzyl)-indoles and indolines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1985-10-30 EP disclosed
US-4532333-A ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1985-07-30 US disclosed
US-4448784-A 1-(Aminoalkylphenyl and aminoalkylbenzyl)-indoles and indolines and analgesic method of use thereof HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1984-05-15 US disclosed
US-4377699-A REACTING INDOLINE WITH AN ORGANIC CARBOXYLIC ACID ACYLATING AGENT, CHLORINATION, SAPONIFICATION, FOLLOWED BY OXIDATION WITH AN AROMATIC NITRO COMPOUND RUTGERSWERKE AKTIENGESELLSCHAFT (DE) 1983-03-22 US disclosed
EP-0004494-B1 DERIVATIVES OF 1,3-DIHYDRO-3-(1-(2-(2,3-DIHYDRO-1,4-BENZODIOXIN-2-YL)2-HYDROXYETHYL)PIPERIDIN-4-YL)2H-INDOL-2-ON, PROCESS FOR THEIR PREPARATION, THEIR USE AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1982-02-17 EP disclosed
EP-0004494-A1 Derivatives of 1,3-dihydro-3-(1-(2-(2,3-dihydro-1,4-benzodioxin-2-yl)2-hydroxyethyl)piperidin-4-yl)2H-indol-2-on, process for their preparation, their use as medicaments and pharmaceutical compositions containing them ROUSSEL-UCLAF (FR) 1979-10-03 EP disclosed
US-4017484-A Cationic dyestuffs BAYER AKTIENGESELLSCHAFT (DT) 1977-04-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250122152-A1 KAT6 Inhibitors KAT6A, KAT6B, KAT7 DRD2 4083/4885DRD4 3715/4885PDE3B 3902/4885
US-20190127345-A1 NEGATIVE PHOTOCHROMIC MATERIALS WITH TUNABLE PROPERTIES ALKBH2, YTHDF2, ANXA2 DRD2 302/4885DRD4 155/4885PDE3B 2944/4885
US-20250109122-A1 CYCLOALKYL PYRIMIDINES AS FERROPORTIN INHIBITORS HAMP, SLC40A1, FANCI DRD2 3430/4885DRD4 3932/4885PDE3B 2809/4885
US-12599584-B2 Indoline derivatives, compositions comprising them and uses thereof IL6, TNF, IDO1 DRD2 1142/4885DRD4 1750/4885PDE3B 840/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.