SCHEMBL5743320

SCHEMBL5743320

O=C(O)CN(Cc1cccc(F)c1)S(=O)(=O)C1(c2cccc3c2oc2ccccc23)C=CC(c2ccccc2)=CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.35
TAS2R14 Q9NYV8 3/20 0.35
DAGLA Q9Y4D2 3/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KCNH2 Q12809 1/20 0.34
SCD5 Q86SK9 1/20 0.33
PER2 O15055 1/20 0.32
CRY1 Q16526 1/20 0.32
CRY2 Q49AN0 1/20 0.32
PTPN2 P17706 1/20 0.32
PTPN1 P18031 1/20 0.32
PTPN6 P29350 1/20 0.32
DUSP3 P51452 1/20 0.32
PTPN11 Q06124 1/20 0.32
PTPN22 Q9Y2R2 1/20 0.32
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5743849 0.87 TAS2R14 (0.35) KEAP1TAS2R14DAGLACYP3A4CYP2D6
SCHEMBL5743318 0.77 KEAP1 (0.37) KEAP1TAS2R14DAGLAPER2CRY1
SCHEMBL5743012 0.76 PTPN1 (0.35) KEAP1DAGLACYP3A4CYP2D6CYP2C9
SCHEMBL4458190 0.71 TAS2R14 (0.51) KEAP1TAS2R14DAGLACYP3A4CYP2D6
SCHEMBL5767369 0.71 MMP12 (0.36) ALDH1A1ALOX5
SCHEMBL4267918 0.70 PTPN1 (0.36) SCD5PTPN1DUSP3
SCHEMBL5744684 0.67 ALOX5 (0.32) ALOX5
SCHEMBL5743846 0.66 TAS2R14 (0.36) KEAP1TAS2R14DAGLAPER2CRY1
SCHEMBL4260729 0.65 PTPN1 (0.35) PTPN1DUSP3ALDH1A1
SCHEMBL4267881 0.64 PTPN1 (0.34) PTPN1DUSP3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006525365-A 2006-11-09 JP claimed
EP-1620422-A2 PHENYL SUBSTITUTED CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B The Institutes for Pharmaceutical Discovery, LLC (US) 2006-02-01 EP claimed
WO-2004099170-A2 PHENYL SUBSTITUTED CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2004-11-18 WO claimed