SCHEMBL5776042

SCHEMBL5776042

CN(C)CC(=C=O)c1cccc(CN(C)C)c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.42
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
ROCK2 O75116 6/20 0.40
HSD17B1 P14061 2/20 0.40
HSD17B2 P37059 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
MEP1B Q16820 5/20 0.38
MEP1A Q16819 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP3A4 P08684 2/20 0.37
PPARG P37231 1/20 0.36
HTR7 P34969 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5779568 0.90 BCHE (0.43) HSD17B1HSD17B2MEP1BMEP1APPARG
SCHEMBL5779117 0.81 MEP1B (0.41) NOS1KMT2AMEN1MEP1BPPARG
SCHEMBL5489563 0.79 HPGD (0.45) ALDH1A1
SCHEMBL5777797 0.79 PBRM1 (0.42) ALDH1A1KMT2AMEN1CYP3A4
SCHEMBL5200753 0.79 PARP1 (0.43) ALDH1A1TSHRKMT2AMEN1L3MBTL1
SCHEMBL289811 0.78 EGFR (0.50) ALDH1A1KMT2A
SCHEMBL5771539 0.76 CES2 (0.50) ALDH1A1KMT2AMEN1
SCHEMBL29630981 0.75 FOLH1 (0.59) ALDH1A1TSHRKMT2AMEN1MEP1B
SCHEMBL168738 0.75 FOLH1 (0.59) ALDH1A1TSHRKMT2AMEN1MEP1B
SCHEMBL3694401 0.75 NOS1 (0.51) NOS1ALDH1A1TSHRROCK2HSD17B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1648875-A1 2-AMINOPHENYL-4-PHENYLPYRIMIDINES AS KINASE INHIBITORS Cyclacel Limited (GB) 2006-04-26 EP disclosed
WO-2005012262-A1 2-AMINOPHENYL-4-PHENYLPYRIMIDINES AS KINASE INHIBITORS CYCLACEL LIMITED (GB) 2005-02-10 WO disclosed