SCHEMBL5845241

SCHEMBL5845241

Cc1ccc(S(=O)(=O)OCC2COc3ccccc3O2)cc1

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.64
SMN1; SMN2 Q16637 2/20 0.60
RAB9A P51151 1/20 0.51
CA2 P00918 4/20 0.49
POLB P06746 1/20 0.48
L3MBTL1 Q9Y468 3/20 0.47
ALDH1A1 P00352 1/20 0.46
MAPK1 P28482 1/20 0.45
MTNR1A P48039 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL567428 1.00 LMNA (0.64) LMNASMN1; SMN2RAB9ACA2POLB
SCHEMBL440397 1.00 LMNA (0.64) LMNASMN1; SMN2RAB9ACA2POLB
SCHEMBL6973472 0.88 CA2 (0.57) LMNASMN1; SMN2RAB9ACA2ALDH1A1
SCHEMBL10832816 0.88 CA2 (0.51) LMNASMN1; SMN2RAB9ACA2ALDH1A1
SCHEMBL6973466 0.88 CA2 (0.57) LMNASMN1; SMN2RAB9ACA2ALDH1A1
SCHEMBL7966432 0.87 LMNA (0.61) LMNASMN1; SMN2RAB9ACA2POLB
SCHEMBL11102654 0.87 LMNA (0.48) LMNASMN1; SMN2RAB9ACA2ALDH1A1
SCHEMBL6976444 0.86 LMNA (0.48) LMNASMN1; SMN2RAB9ACA2POLB
SCHEMBL6976439 0.86 LMNA (0.48) LMNASMN1; SMN2RAB9ACA2POLB
SCHEMBL7782073 0.86 LMNA (0.48) LMNASMN1; SMN2RAB9ACA2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-8325260-A None JP disclosed
EP-3233077-B1 DOPAMINE D2 RECEPTOR LIGANDS BROAD INST INC (US) 2026-05-06 EP disclosed
US-12428373-B2 Dopamine D2 receptor ligands THE BROAD INSTITUTE, INC. (US) 2025-09-30 US disclosed
US-20230143552-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2023-05-11 US disclosed
US-11498896-B2 Dopamine D2 receptor ligands THE BROAD INSTITUTE, INC. (US) 2022-11-15 US disclosed
US-20210147355-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2021-05-20 US disclosed
US-10633336-B2 Dopamine D2 receptor ligands THE BROAD INSTITUTE, INC. (US) 2020-04-28 US disclosed
US-20190152992-A1 BENZODIOXANE DERIVATIVES AND THEIR PHARMACEUTICAL USE ORION CORPORATION (FI) 2019-05-23 US disclosed
US-20180155283-A1 DOPAMINE D2 RECEPTOR LIGANDS THE BROAD INSTITUTE, INC. (US) 2018-06-07 US disclosed
EP-3233077-A1 DOPAMINE D2 RECEPTOR LIGANDS The Broad Institute Inc. (US) 2017-10-25 EP disclosed
US-4826848-A Antidepressive substituted N-[(4-piperidinyl)alkyl] bicyclic condensed oxazol- and thiazolamines JANSSEN PHARMACEUTICA N.V. (BE) 1989-05-02 US disclosed
US-4749702-A PARKINSON*S DISEASE, ENTEROKINESIA JANSSEN PHARMACEUTICA N. V. (BE) 1988-06-07 US disclosed
US-4702763-A Herbicidal 1-aryl-delta2-1,2,4-triazolin-5-ones FMC CORPORATION (US) 1987-10-27 US disclosed
US-4689330-A PARKINSON DISEASE JANSSEN PHARMACEUTICA N.V. (BE) 1987-08-25 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed
EP-0199400-A2 Substituted N-[(4-piperidinyl)alkyl] bicyclic condensed ozazol- and thiazolamines JANSSEN PHARMACEUTICA N.V. (BE) 1986-10-29 EP disclosed
US-4579845-A Antihypertensive cyanoguanidines BOUCHARA S.A. (FR) 1986-04-01 US disclosed
EP-0157876-A1 HERBICIDAL 1-ARYL-$g(D)?2 -1,2,4-TRIAZOLIN-5-ONES FMC Corporation (US) 1985-10-16 EP disclosed
WO-1985001637-A1 HERBICIDAL 1-ARYL-DELTA2-1,2,4-TRIAZOLIN-5-ONES FMC CORPORATION (US) 1985-04-25 WO disclosed
US-4470989-A Neuroleptic n-oxacyclyl-alkylpiperidine derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1984-09-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180155283-A1 DOPAMINE D2 RECEPTOR LIGANDS DRD2, DRD3, ARRB1 LMNA 4642/4885SMN1; SMN2 2087/4885RAB9A 889/4885
US-11498896-B2 Dopamine D2 receptor ligands DRD2, SLC6A3, NTSR2 LMNA 4865/4885SMN1; SMN2 1443/4885RAB9A 906/4885
US-10633336-B2 Dopamine D2 receptor ligands DRD2, ARRB1, DRD3 LMNA 4825/4885SMN1; SMN2 2679/4885RAB9A 920/4885
US-20230143552-A1 DOPAMINE D2 RECEPTOR LIGANDS DRD2, SLC6A3, NTSR2 LMNA 4865/4885SMN1; SMN2 1443/4885RAB9A 906/4885
US-20210147355-A1 DOPAMINE D2 RECEPTOR LIGANDS DRD2, SLC6A3, NTSR2 LMNA 4865/4885SMN1; SMN2 1443/4885RAB9A 906/4885
US-12428373-B2 Dopamine D2 receptor ligands DRD2, SLC6A3, NTSR2 LMNA 4865/4885SMN1; SMN2 1443/4885RAB9A 906/4885
US-20190152992-A1 BENZODIOXANE DERIVATIVES AND THEIR PHARMACEUTICAL USE TBXA2R, ADRA2C, ADRB2 LMNA 2674/4885SMN1; SMN2 1954/4885RAB9A 2884/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.