SCHEMBL5859873

SCHEMBL5859873

COC1=C(OC)C(=O)C(c2cc(C)c(-c3ccncc3)c(C(=O)NC3CCCCC3)c2)=C(C)C1=O

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 6/20 0.50
CNR2 P34972 6/20 0.50
RAB9A P51151 4/20 0.42
NPC1 O15118 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ALDH1A1 P00352 4/20 0.41
HTT P42858 1/20 0.41
ROCK2 O75116 3/20 0.41
ROCK1 Q13464 1/20 0.41
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HPGD P15428 3/20 0.39
BACE1 P56817 1/20 0.39
KDM4E B2RXH2 2/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6655451 0.99 CNR1 (0.48) CNR1CNR2RAB9ANPC1L3MBTL1
SCHEMBL5859140 0.95 CNR1 (0.45) CNR1CNR2ROCK2ROCK1
SCHEMBL5859860 0.81 IKBKB (0.37) KDM4E
SCHEMBL5862246 0.80 CYP2C9 (0.41) RAB9AALDH1A1HTTMEN1KMT2A
SCHEMBL5859281 0.79 CYP3A4 (0.48) RAB9ANPC1ALDH1A1MEN1KMT2A
SCHEMBL5859286 0.79 TAS1R3 (0.38) CNR2ALDH1A1HTTROCK2ROCK1
SCHEMBL5860337 0.77 APOB (0.44)
SCHEMBL5859258 0.75 ALDH1A1 (0.40) RAB9ANPC1L3MBTL1ALDH1A1HTT
SCHEMBL5859099 0.74 CNR2 (0.42) CNR1CNR2RAB9AL3MBTL1ALDH1A1
SCHEMBL5862115 0.73 ROCK2 (0.41) CNR1CNR2RAB9AL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7122543-B2 Substituted benzoic acid derivatives having NF-κB inhibiting action DAIICHI SUNTORY PHARMA CO., LTD. (JP) 2006-10-17 US disclosed
EP-1437339-A1 SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING NF-KAPPA B INHIBITING ACTIVITY Daiichi Suntory Pharma Co., Ltd. (JP) 2004-07-14 EP disclosed