SCHEMBL6655451

SCHEMBL6655451

COC1=C(OC)C(=O)C(c2cc(C)c(-c3ccncc3)c(C(=O)NC3CCCC3)c2)=C(C)C1=O

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 7/20 0.48
CNR2 P34972 7/20 0.48
ROCK2 O75116 4/20 0.41
ROCK1 Q13464 1/20 0.41
RAB9A P51151 3/20 0.41
NPC1 O15118 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HTT P42858 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5859873 0.99 CNR1 (0.50) CNR1CNR2ROCK2ROCK1RAB9A
SCHEMBL5859140 0.96 CNR1 (0.45) CNR1CNR2ROCK2ROCK1
SCHEMBL5859860 0.82 IKBKB (0.37) MAPT
SCHEMBL5859281 0.80 CYP3A4 (0.48) RAB9ANPC1ALDH1A1MAPT
SCHEMBL5859286 0.80 TAS1R3 (0.38) CNR2ROCK2ROCK1HTTALDH1A1
SCHEMBL5862246 0.79 CYP2C9 (0.41) RAB9AHTTALDH1A1
SCHEMBL5860337 0.78 APOB (0.44)
SCHEMBL5859258 0.76 ALDH1A1 (0.40) RAB9ANPC1L3MBTL1HTTALDH1A1
SCHEMBL5862115 0.73 ROCK2 (0.41) CNR1CNR2ROCK2ROCK1RAB9A
SCHEMBL5859099 0.73 CNR2 (0.42) CNR1CNR2ROCK2RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1437339-A1 SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING NF-KAPPA B INHIBITING ACTIVITY Daiichi Suntory Pharma Co., Ltd. (JP) 2004-07-14 EP disclosed