SCHEMBL6047645

SCHEMBL6047645

Cc1ccc(C2=C(Cl)C(Cl)=C(c3ccccc3C(F)(F)F)[CH]C2)cc1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 11/20 0.38
TRPA1 O75762 3/20 0.35
AR P10275 1/20 0.34
TRPM8 Q7Z2W7 1/20 0.34
CRHR1 P34998 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887436 0.81 CYP2A6 (0.36) HSD11B1
SCHEMBL6047589 0.77 PTGS1 (0.35)
SCHEMBL1047574 0.74 HSD11B1 (0.52) HSD11B1TRPA1ARTRPM8
SCHEMBL6047588 0.73 NPBWR1 (0.38) HSD11B1
SCHEMBL28922699 0.72 HSD11B1 (0.50) HSD11B1TRPA1ARTRPM8
SCHEMBL5887404 0.71 L3MBTL1 (0.40)
SCHEMBL6047653 0.71 HSD11B1 (0.37) HSD11B1
SCHEMBL5887582 0.64 TSHR (0.43)
SCHEMBL22304414 0.64 AR (0.58) HSD11B1TRPA1ARTRPM8
SCHEMBL24297565 0.62 AR (0.56) HSD11B1TRPA1ARTRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed