Hexoprenaline

Hexoprenaline

SCHEMBL598186

O=S(=O)(O)O.Oc1ccc(C(O)CNCCCCCCNCC(O)c2ccc(O)c(O)c2)cc1O

nearest known ligand 0.88

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3CALCRLCHRM1CHRM2CHRM3F2RMAOAMAOBMAP2K1MAP2K2NTRK1NTRK2NTRK3OPRD1OPRK1OPRM1P2RY12PKLRSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASLC18A2SLC6A2SLC6A3TLR7TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8dacAdacBdacCfolAftsImrcAmrcBmrdApolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmB1rpmB2rpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmHrpmIrpmJrpmJ2rpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsR1rpsR2rpsSrpsTrpsUrpsZykgMykgO

The experimentally established mechanism targets of Hexoprenaline. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 known ✓ P07550 12/20 0.65
ADRB1 known ✓ P08588 8/20 0.55
ADRB3 known ✓ P13945 5/20 0.55
ADRA1D known ✓ P25100 2/20 0.55
ADRA1A known ✓ P35348 2/20 0.55
ADRA1B known ✓ P35368 2/20 0.55
ADRA2A known ✓ P08913 1/20 0.55
ADRA2B known ✓ P18089 1/20 0.55
ADRA2C known ✓ P18825 1/20 0.55
SLC6A2 known ✓ P23975 1/20 0.50
MAPT P10636 5/20 0.55
TDP1 Q9NUW8 5/20 0.55
KDM4E B2RXH2 5/20 0.55
DRD2 P14416 4/20 0.55
DRD3 P35462 4/20 0.55
HSD17B10 Q99714 4/20 0.55
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
MTOR P42345 3/20 0.55
TSHR P16473 3/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hexoprenaline SCHEMBL121449 0.94 ADRB2 (0.72) ADRB2ADRB1MAPTTDP1KDM4E
Hexoprenaline SCHEMBL32668781 0.94 ADRB2 (0.72) ADRB2ADRB1MAPTTDP1KDM4E
Hexoprenaline SCHEMBL1604446 0.92 ADRB2 (0.70) ADRB2ADRB1MAPTTDP1KDM4E
Hexoprenaline SCHEMBL3500862 0.92 ADRB2 (0.70) ADRB2ADRB1MAPTTDP1KDM4E
SCHEMBL8442887 0.87 ADRB2 (0.63) ADRB2ADRB1MAPTTDP1KDM4E
SCHEMBL9768151 0.87 ADRB2 (0.63) ADRB2ADRB1MAPTTDP1KDM4E
SCHEMBL9768158 0.87 ADRB2 (0.63) ADRB2ADRB1MAPTTDP1KDM4E
SCHEMBL31530707 0.85 ADRB2 (0.68) ADRB2ADRB1MAPTTDP1KDM4E
SCHEMBL31530706 0.85 ADRB2 (0.68) ADRB2ADRB1MAPTTDP1KDM4E
SCHEMBL13790391 0.85 ADRB2 (0.62) ADRB2ADRB1MAPTTDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 487 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 US claimed
US-8263125-B2 Dosage form for high dose-high solubility active ingredients that provides for immediate release and modified release of the active ingredients TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-11 US claimed
US-20060024365-A1 Novel dosage form VAYA NAVIN 2006-02-02 US claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
EP-0580860-B2 METHOD OF MANUFACTURING SOLID DISPERSION NIPPON SHINYAKU CO LTD (JP) 2004-12-15 EP claimed
US-5811547-A Method for inducing crystalline state transition in medicinal substance NIPPON SHINYAJU CO., LTD. (JP) 1998-09-22 US claimed
US-5700410-A Method of manufacturing wax matrices NIPPON SHINYAKU CO., LTD. (JP) 1997-12-23 US claimed
EP-0580860-B1 METHOD OF MANUFACTURING SOLID DISPERSION NIPPON SHINYAKU CO LTD (JP) 1997-10-22 EP claimed
US-12629379-B2 Pharmaceutical composition for preventing, suppressing, or treating symptom associated with allergic reaction NIPPON CHEMIPHAR CO., LTD. (JP) 2026-05-19 US disclosed
EP-4706683-A2 CHEWABLE FORMULATIONS Elanco Tiergesundheit AG (CH) 2026-03-11 EP disclosed
US-20260034059-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES AQUESTIVE THERAPEUTICS, INC. (US) 2026-02-05 US disclosed
US-20260000678-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING, SUPPRESSING, OR TREATING SYMPTOM ASSOCIATED WITH PSEUDO-ALLERGIC REACTION TAKASAKI UNIV OF HEALTH AND WELFARE (JP) 2026-01-01 US disclosed
US-12465564-B2 Oral and nasal compositions and methods of treatment AQUESTIVE THERAPEUTICS, INC. (US) 2025-11-11 US disclosed
US-4801458-A POROUS HOLLOW FIBERS FILLED WITH MEDICINE TEIJIN LIMITED (JP) 1989-01-31 US disclosed
US-4755544-A Sustained release preparation TEIJIN LIMITED (JP) 1988-07-05 US disclosed
EP-0253901-A1 SUSTAINED-RELEASE PREPARATION TEIJIN LIMITED (JP) 1988-01-27 EP disclosed
EP-0227836-A1 SUSTAINED RELEASING PATCH TEIJIN LIMITED (JP) 1987-07-08 EP disclosed
EP-0207638-A2 Sustained-release pharmaceutical preparation TEIJIN LIMITED (JP) 1987-01-07 EP disclosed
EP-0187703-A2 Sustained release preparation TEIJIN LIMITED (JP) 1986-07-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12629379-B2 Pharmaceutical composition for preventing, suppressing, or treating symptom associated with allergic reaction HRH2, HRH4, HRH1 ADRB2 39/4885ADRB1 43/4885ADRB3 66/4885
US-20260000678-A1 PHARMACEUTICAL COMPOSITION FOR PREVENTING, SUPPRESSING, OR TREATING SYMPTOM ASSOCIATED WITH PSEUDO-ALLERGIC REACTION TRPV1, TRPV4, TRPV5 ADRB2 537/4885ADRB1 503/4885ADRB3 382/4885
US-20260034059-A1 ORAL FILM COMPOSITIONS AND DOSAGE FORMS HAVING PRECISE ACTIVE DISSOLUTION PROFILES SORD, SLC6A13, CACNA1A ADRB2 2249/4885ADRB1 2529/4885ADRB3 2864/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.