SCHEMBL6023749

SCHEMBL6023749

CC(C)Cc1cc2ccccc2c(CC(C)C)c1S(=O)(=O)[O-].[Na+]

nearest known ligand 0.36

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR3C1 known ✓ P04150 1/20 0.32
GPR35 Q9HC97 1/20 0.34
HTR2A P28223 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ENTPD1 P49961 1/20 0.33
ENTPD2 Q9Y5L3 1/20 0.33
PTGER1 P34995 1/20 0.33
NR1I2 O75469 1/20 0.33
PGR P06401 1/20 0.32
NR3C2 P08235 1/20 0.32
SLC2A1 P11166 1/20 0.32
GPR84 Q9NQS5 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ATM Q13315 1/20 0.31
ELANE P08246 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29460462 0.89 NR1I2 (0.35) GPR35ENTPD1ENTPD2PTGER1NR1I2
SCHEMBL37571 0.89 NR1I2 (0.35) GPR35ENTPD1ENTPD2PTGER1NR1I2
Potassium Ion SCHEMBL23749083 0.86 NR1I2 (0.33) HTR2AL3MBTL1ENTPD1ENTPD2PTGER1
SCHEMBL6555708 0.84 CYP2D6 (0.40) GPR35HTR2AL3MBTL1NR3C1PGR
SCHEMBL27345267 0.83 CYP2D6 (0.40) GPR35HTR2AL3MBTL1NR3C1PGR
SCHEMBL1024286 0.78 NR1I2 (0.35) HTR2APTGER1NR1I2NR3C1PGR
Sulfuric Acid SCHEMBL28020160 0.78 MAPT (0.38) HTR2APTGER1SLC2A1KDM4E
SCHEMBL10790517 0.77 HTR2A (0.42) HTR2AL3MBTL1GPR84KDM4EATM
SCHEMBL29720 0.76 CYP2D6 (0.43) NR3C1PGRNR3C2SLC2A1GPR84
SCHEMBL29364308 0.76 CYP2D6 (0.43) NR3C1PGRNR3C2SLC2A1GPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7101900-B2 Benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides BASF AKTIENGESELLSCHAFT (DE) 2006-09-05 US disclosed
US-20050187265-A1 Novel benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides RHEINHEIMER JOACHIM (DE) 2005-08-25 US disclosed
US-6881742-B1 Benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides BASF AKTIENGESELLSCHAFT (DE) 2005-04-19 US disclosed
US-6680402-B2 SUCH AS N-PHENYLACETYL-2-DIFLUOROMETHOXY-6-FLUOROBENZAMIDE-O-CYCLOPROPYLMETHYL OXIME BASF AKTIENGESELLSCHAFT (DE) 2004-01-20 US disclosed
US-6680283-B1 TREATMENT OF PLANTS, AND ALSO FOR THE THERAPEUTIC TREATMENT OF HUMAN DISORDERS CAUSED BY HARMFUL FUNGI, AND FOR THE VETERINARY TREATMENT OF MAMMALS BASF AKTIENGESELLSCHAFT (DE) 2004-01-20 US disclosed
US-6586369-B1 Agriculture BASF AKTIENGESELLSCHAFT (DE) 2003-07-01 US disclosed
US-20030120085-A1 Novel benzamidoxime derivatives, intermediates and processes for their preparation, and their use as fungicides EICKEN KARL (DE) 2003-06-26 US disclosed
US-6509501-B2 Agriculture BASF AKTIENGESELLSCHAFT (DE) 2003-01-21 US disclosed
US-6476061-B1 Fungicides containing pyrrolidones as their active agents BASF AKTIENGESELLSCHAFT (DE) 2002-11-05 US disclosed
US-20020133025-A1 Novel benzamidoxime derivatives, intermediates and processes for their preparation, and their use as fungicides EICKEN KARL (DE) 2002-09-19 US disclosed
US-6420605-B1 DIFLUOROMETHYL ETHERS OF BENZAMIDOXIME COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-07-16 US disclosed
US-6417398-B1 Benzamidoxim derivatives, intermediate products and methods for preparing them, and their use as fungicides BASF AKTIENGESELLSCHAFT (DE) 2002-07-09 US disclosed
US-6147104-A USED IN COMBATING PARASITIC FUNGUS BASF AKTIENGESELLSCHAFT (DE) 2000-11-14 US disclosed
US-5998450-A FOR PLANTS BASF AKTIENGESELLSCHAFT (DE) 1999-12-07 US disclosed
US-5922899-A Carbamoyl carboxylic acid amides BASF AKTIENGESELLSCHAFT (DE) 1999-07-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020133025-A1 Novel benzamidoxime derivatives, intermediates and processes for their preparation, and their use as fungicides CBR1, CBR3, CYP1B1 NR3C1 1861/4885GPR35 3061/4885HTR2A 3815/4885
US-20050187265-A1 Novel benzyl amidoxime derivatives, intermediate products and method for their production and use as fungicides CBR3, CBR1, CYP1B1 NR3C1 1218/4885GPR35 3455/4885HTR2A 2326/4885
US-20030120085-A1 Novel benzamidoxime derivatives, intermediates and processes for their preparation, and their use as fungicides CBR1, CBR3, CYP1B1 NR3C1 1861/4885GPR35 3061/4885HTR2A 3815/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.