SCHEMBL6047653

SCHEMBL6047653

Cc1ccc(C2=C(Cl)C(Cl)=C(c3cccc(OC(F)(F)F)c3)[CH]C2)cc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.37
DRD2 P14416 1/20 0.36
DRD1 P21728 1/20 0.36
PTGES2 Q9H7Z7 1/20 0.36
DHODH Q02127 4/20 0.36
PDE10A Q9Y233 1/20 0.36
GPR3 P46089 1/20 0.36
GALR1 P47211 1/20 0.36
S1PR1 P21453 1/20 0.35
SLC5A1 P13866 2/20 0.35
KCNH2 Q12809 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35
MMP2 P08253 1/20 0.35
MMP3 P08254 1/20 0.35
CCKAR P32238 1/20 0.35
CYP1A2 P05177 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C19 P33261 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047588 0.86 NPBWR1 (0.38) HSD11B1GPR3MAPT
SCHEMBL5887570 0.85 ALKBH3 (0.44) CCKARCYP1A2MAPTCYP2C19
SCHEMBL5887404 0.81 L3MBTL1 (0.40) MAPT
SCHEMBL5887672 0.79 ESR2 (0.40)
SCHEMBL1044062 0.76 CYP1A2 (0.51) PTGES2DHODHGPR3GALR1S1PR1
SCHEMBL5887443 0.72 ACHE (0.46) MAPT
SCHEMBL5887582 0.72 TSHR (0.43) MMP2MAPT
SCHEMBL6047589 0.69 PTGS1 (0.35) DHODH
SCHEMBL5542229 0.68 PTGES2 (0.50) HSD11B1PTGES2DHODHGPR3GALR1
SCHEMBL278095 0.68 GPR3 (0.48) PTGES2DHODHPDE10AGPR3GALR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed