SCHEMBL6050489

SCHEMBL6050489

CON(C)C(=O)c1ccon1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.37
CHRNA4 P43681 2/20 0.36
CLK1 P49759 1/20 0.35
DYRK1A Q13627 1/20 0.35
DYRK1B Q9Y463 1/20 0.35
TRPM8 Q7Z2W7 2/20 0.35
PSMB8 P28062 2/20 0.34
RAB9A P51151 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PKM P14618 1/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
RAPGEF3 O95398 1/20 0.32
RAPGEF4 Q8WZA2 1/20 0.32
SLC6A3 Q01959 1/20 0.32
NPC1 O15118 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2362735 0.81 CHRNA4 (0.39) CHRNA4RAB9AMEN1KMT2AALDH1A1
SCHEMBL17611640 0.76 PSMB8 (0.30) CHRNA4PSMB8
SCHEMBL17611638 0.76 PSMB8 (0.30) CHRNA4PSMB8
SCHEMBL11722748 0.75 CHRNA4 (0.36) CHRNA4RAB9AALDH1A1L3MBTL1RAPGEF3
SCHEMBL26269687 0.74 PSMB8 (0.39) MLYCDCHRNA4PSMB8RAB9AMEN1
SCHEMBL7261615 0.73 PSMB8 (0.36) CHRNA4PSMB8RAB9AACACB
SCHEMBL2122427 0.73
SCHEMBL28399251 0.73 ALDH1A1 (0.50) MLYCDRAB9ATDP1ALDH1A1L3MBTL1
SCHEMBL19456683 0.72 RECQL (0.36) CHRNA4PSMB8RAB9AMEN1KMT2A
SCHEMBL8374791 0.72 KDM4E (0.45) MLYCDCLK1DYRK1ADYRK1BTRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 127 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3829559-B1 INHIBITORS OF HISTONE DEACETYLASE USEFUL FOR THE TREATMENT OR PREVENTION OF HIV INFECTION MERCK SHARP & DOHME LLC (US) 2026-05-13 EP disclosed
US-20260103457-A1 NOVEL PROCESS FOR PREPARATION OF SOLUBLE GUANYLATE CYCLASE STIMULATORS CYCLERION THERAPEUTICS INC (US) 2026-04-16 US disclosed
US-20250361228-A1 PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF SOLUBLE GUANYLATE CYCLASE STIMULATORS CYCLERION THERAPEUTICS INC (US) 2025-11-27 US disclosed
US-20250255821-A1 SOLID DISPERSIONS COMPRISING A SGC STIMULATOR CYCLERION THERAPEUTICS, INC. 2025-08-14 US disclosed
US-12365674-B2 Inhibitors of histone deacetylase useful for the treatment or prevention of HIV infection MERCK SHARP & DOHME LLC (US) 2025-07-22 US disclosed
EP-4570797-A2 NOVEL PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF SOLUBLE GUANYLATE CYCLASE STIMULATORS Cyclerion Therapeutics, Inc. (US) 2025-06-18 EP disclosed
US-12331044-B2 Inhibitors of histone deacetylase useful for the treatment or prevention of HIV infection MERCK SHARP & DOHME LLC (US) 2025-06-17 US disclosed
US-20250129060-A1 SOLID FORMS OF AN SGC STIMULATOR CYCLERION THERAPEUTICS INC (US) 2025-04-24 US disclosed
US-12275724-B2 Processes and intermediates for the preparation of soluble guanylate cyclase stimulators CYCLERION THERAPEUTICS, INC. (US) 2025-04-15 US disclosed
US-20250109126-A1 DIHYDRO-OXAZOL DERIVATIVE COMPOUNDS AC IMMUNE SA (CH) 2025-04-03 US disclosed
WO-2016044447-A1 PYRAZOLE DERIVATIVES AS SGC STIMULATORS IRONWOOD PHARMACEUTICALS, INC. (US) 2016-03-24 WO disclosed
EP-1414802-B1 HETEROARYLHETEROALKYLAMINE DERIVATIVES AND THEIR USE AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2006-04-26 EP disclosed
US-6887871-B2 Use of phenylheteroakylamine derivatives ASTRAZENECA AB (SE) 2005-05-03 US disclosed
EP-1263711-B1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2004-12-15 EP disclosed
US-20040176422-A1 Heteroarylheteroalkylamine derivatives and their use as inhibitors of nitric oxide synthase ASTRAZENECA AB (SE) 2004-09-09 US disclosed
EP-1414802-A1 HETEROARYLHETEROALKYLAMINE DERIVATIVES AND THEIR USE AS INHIBITORS OF NITRIC OXIDE SYNTHASE AstraZeneca AB (SE) 2004-05-06 EP disclosed
US-20030158185-A1 Novel use of phenylheteroakylamine derivatives ASTRAZENECA AB (SE) 2003-08-21 US disclosed
WO-2003011830-A1 HETEROARYLHETEROALKYLAMINE DERIVATIVES AND THEIR USE AS INHIBITORS OF NITRIC OXIDE SYNTHASE ASTRAZENECA AB (SE) 2003-02-13 WO disclosed
EP-1263711-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP disclosed
WO-2001062704-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12275724-B2 Processes and intermediates for the preparation of soluble guanylate cyclase stimulators GUCY1A2, GUCY1B1, GUCY1B2 MLYCD 607/4885CHRNA4 1900/4885CLK1 3805/4885
US-12331044-B2 Inhibitors of histone deacetylase useful for the treatment or prevention of HIV infection HDAC1, HDAC11, HDAC10 MLYCD 4011/4885CHRNA4 4013/4885CLK1 4539/4885
US-20250361228-A1 PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF SOLUBLE GUANYLATE CYCLASE STIMULATORS GUCY1A2, GUCY1B1, GUCY1B2 MLYCD 607/4885CHRNA4 1900/4885CLK1 3805/4885
US-20250255821-A1 SOLID DISPERSIONS COMPRISING A SGC STIMULATOR GMPS, PRKG1, GUCY1A2 MLYCD 1621/4885CHRNA4 1547/4885CLK1 3029/4885
US-12365674-B2 Inhibitors of histone deacetylase useful for the treatment or prevention of HIV infection HDAC1, HDAC11, HDAC3 MLYCD 4125/4885CHRNA4 3226/4885CLK1 4195/4885
US-20250129060-A1 SOLID FORMS OF AN SGC STIMULATOR GUCY1A2, PRKG1, GUCY1A1 MLYCD 1240/4885CHRNA4 2571/4885CLK1 2798/4885
US-20040176422-A1 Heteroarylheteroalkylamine derivatives and their use as inhibitors of nitric oxide synthase NOS3, NOS1, NOS2 MLYCD 4272/4885CHRNA4 1294/4885CLK1 965/4885
US-20250109126-A1 DIHYDRO-OXAZOL DERIVATIVE COMPOUNDS NLRP3, NLRP1, NOD1 MLYCD 639/4885CHRNA4 4247/4885CLK1 3230/4885
US-20260103457-A1 NOVEL PROCESS FOR PREPARATION OF SOLUBLE GUANYLATE CYCLASE STIMULATORS GUCY1B1, GUCY1B2, GUCY1A2 MLYCD 1033/4885CHRNA4 2129/4885CLK1 2771/4885
US-20030158185-A1 Novel use of phenylheteroakylamine derivatives NOS1, XDH, NOS2 MLYCD 2885/4885CHRNA4 1794/4885CLK1 1637/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.