SCHEMBL6074907

SCHEMBL6074907

CCOC(=O)C(C(=O)OCC)c1ccccc1N

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.54
HSD17B10 Q99714 3/20 0.54
MMP8 P22894 1/20 0.53
PIN1 Q13526 1/20 0.45
TSHR P16473 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
MEN1 O00255 2/20 0.44
NPC1 O15118 2/20 0.44
KMT2A Q03164 2/20 0.44
CASP1 P29466 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAOA P21397 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CDC25B P30305 2/20 0.40
POLB P06746 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28996258 0.85 ALDH1A1 (0.56) ALDH1A1HSD17B10MMP8TSHRKMT2A
SCHEMBL7509738 0.81 MMP8 (0.51) ALDH1A1HSD17B10MMP8PIN1TSHR
SCHEMBL11514512 0.80 ALDH1A1 (0.49) ALDH1A1HSD17B10MMP8PIN1TSHR
SCHEMBL1044283 0.80 NLRP3 (0.50) ALDH1A1MMP8PIN1TSHRMEN1
SCHEMBL7513221 0.80 MMP8 (0.50) ALDH1A1HSD17B10MMP8PIN1TSHR
SCHEMBL27618923 0.79 ALDH1A1 (0.47) ALDH1A1HSD17B10MMP8PIN1TSHR
SCHEMBL2003346 0.79 MEN1 (0.50) ALDH1A1MMP8PIN1TSHRMEN1
SCHEMBL5530167 0.79 MMP8 (0.49) ALDH1A1MMP8PIN1TSHRMEN1
SCHEMBL5861445 0.79 CASP1 (0.59) ALDH1A1MMP8PIN1TSHRMEN1
SCHEMBL3414451 0.77 LMNA (0.43) ALDH1A1HSD17B10KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7115784-B2 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2006-10-03 US disclosed
US-6759554-B2 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2004-07-06 US disclosed
US-20040019216-A1 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2004-01-29 US disclosed
US-20030065187-A1 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-04-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030065187-A1 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds ADH5, CBR3, ALDH3A1 ALDH1A1 26/4885HSD17B10 352/4885MMP8 3433/4885
US-20040019216-A1 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds ADH5, CBR3, ALDH3A1 ALDH1A1 26/4885HSD17B10 352/4885MMP8 3433/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.