SCHEMBL6089139

SCHEMBL6089139

Cc1cccc(COc2cccc(OCCOc3ccccn3)c2)c1OCC#N

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.36
CCNB2 O95067 1/20 0.35
CDK1 P06493 1/20 0.35
CDK4 P11802 1/20 0.35
CCNB1 P14635 1/20 0.35
CCND1 P24385 1/20 0.35
CCNB3 Q8WWL7 1/20 0.35
FFAR1 O14842 2/20 0.35
GRM5 P41594 1/20 0.34
MAPT P10636 2/20 0.33
PPARG P37231 1/20 0.33
TP53 P04637 1/20 0.33
HTR1A P08908 2/20 0.33
ADRA1D P25100 2/20 0.33
ADRA1A P35348 2/20 0.33
ADRA1B P35368 2/20 0.33
AURKA O14965 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6091382 0.88 CCNB2 (0.40) SMN1; SMN2CCNB2CDK1CDK4CCNB1
SCHEMBL5725263 0.86 SCN8A (0.38) SMN1; SMN2CCNB2CDK1CDK4CCNB1
SCHEMBL6089925 0.86 ABCB1 (0.42) SMN1; SMN2CCNB2CDK1CDK4CCNB1
SCHEMBL6088697 0.82 PTGDR2 (0.46) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL6090892 0.81 BCHE (0.40) FFAR1NR4A2
SCHEMBL6088303 0.80 NOS3 (0.46) SMN1; SMN2HTTKMT2AMAPK1
SCHEMBL5725097 0.78 CHRNB2 (0.40) CCNB2CDK1CDK4CCNB1CCND1
SCHEMBL6088282 0.78 ALOX5 (0.42) RAB9A
SCHEMBL6092118 0.77 HTR1A (0.44) HTR1ASCN8AMAPK1
SCHEMBL6089251 0.77 SLC26A4 (0.49) CCNB2CDK1CDK4CCNB1CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7005440-B1 Therapeutic uses of tri-aryl acid derivatives AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2006-02-28 US disclosed
EP-1177176-A1 TRI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS Aventis Pharma Deutschland GmbH (DE) 2002-02-06 EP disclosed
WO-2000064876-A1 TRI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-11-02 WO disclosed