SCHEMBL6154538

SCHEMBL6154538

O=Cc1cccc(C(O)c2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.50
PNMT P11086 1/20 0.50
ACP3 P15309 2/20 0.47
IDO1 P14902 1/20 0.44
TDO2 P48775 1/20 0.44
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
MAOB P27338 1/20 0.41
FBP1 P09467 1/20 0.41
POLB P06746 1/20 0.41
HSD17B2 P37059 1/20 0.40
P4HB P07237 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
HSP90AA1 P07900 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
KMT2A Q03164 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4135956 0.85 PNMT (0.65) CES2PNMTACP3IDO1TDO2
SCHEMBL67201 0.81 FBP1 (0.56) CES2ALDH1A1L3MBTL1MAOBFBP1
SCHEMBL29425705 0.81 FBP1 (0.56) CES2ALDH1A1L3MBTL1MAOBFBP1
SCHEMBL4135655 0.80 PNMT (0.59) CES2PNMTACP3IDO1TDO2
SCHEMBL2642178 0.80 UNG (0.48) ALDH1A1L3MBTL1MAOBLMNA
SCHEMBL28376765 0.78 MAOA (0.44) CES2ALDH1A1MAOBMEN1KMT2A
SCHEMBL31067471 0.77 TSHR (0.66) CES2PNMTACP3IDO1TDO2
SCHEMBL17073488 0.77 TSHR (0.66) CES2PNMTACP3IDO1TDO2
SCHEMBL1712441 0.77 PNMT (0.56) CES2PNMTACP3IDO1TDO2
Acetaldehyde SCHEMBL28151033 0.76 NFE2L2 (0.54) CES2ALDH1A1L3MBTL1MAOBFBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050065118-A1 Organosulfur inhibitors of tyrosine phosphatases METABASIS THERAPEUTICS, INC. 2005-03-24 US disclosed
EP-1446110-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES Structural Bioinformatics Inc. (US) 2004-08-18 EP disclosed
WO-2003032916-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES STRUCTURAL BIOINFORMATICS INC. (US) 2003-04-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050065118-A1 Organosulfur inhibitors of tyrosine phosphatases PTPRS, PTPRJ, PTPRCAP CES2 1903/4885PNMT 330/4885ACP3 773/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.