SCHEMBL6167296

SCHEMBL6167296

Cc1nn(-c2ccccc2)c2c1C(=O)CC(C(C)C)C2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.45
ALDH1A1 P00352 2/20 0.45
CCNA2 P20248 2/20 0.45
CDK2 P24941 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
DHODH Q02127 1/20 0.43
TSHR P16473 2/20 0.42
OPRM1 P35372 5/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
LMNA P02545 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
PIK3CD O00329 1/20 0.39
PIK3R1 P27986 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6771481 0.87 OPRM1 (0.43) HIF1ASMN1; SMN2ALDH1A1CCNA2CDK2
SCHEMBL6770476 0.87 OPRM1 (0.45) HIF1ASMN1; SMN2ALDH1A1DHODHOPRM1
SCHEMBL6769819 0.87 OPRM1 (0.43) SMN1; SMN2ALDH1A1MEN1KMT2ADHODH
SCHEMBL6164547 0.86 DHODH (0.43) HIF1ASMN1; SMN2ALDH1A1CCNA2CDK2
SCHEMBL6770505 0.86 OPRM1 (0.46) SMN1; SMN2MEN1KMT2ADHODHOPRM1
SCHEMBL6168419 0.85 DHODH (0.42) HIF1ASMN1; SMN2ALDH1A1CCNA2CDK2
SCHEMBL6164978 0.84 DHODH (0.41) HIF1ASMN1; SMN2ALDH1A1CCNA2CDK2
SCHEMBL6162163 0.83 DHODH (0.41) HIF1ASMN1; SMN2ALDH1A1CCNA2CDK2
SCHEMBL6167870 0.82 ALDH1A1 (0.49) HIF1ASMN1; SMN2ALDH1A1CCNA2CDK2
SCHEMBL6165346 0.82 ALDH1A1 (0.40) HIF1ASMN1; SMN2ALDH1A1CCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed