SCHEMBL6188992

SCHEMBL6188992

Cc1[nH]c2ccc(N)cc2c1C(=O)c1c(F)cccc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
MAPT P10636 1/20 0.41
NGFR P08138 1/20 0.40
GAA P10253 1/20 0.39
PARP1 P09874 1/20 0.39
ALOX15 P16050 1/20 0.39
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
NR4A2 P43354 1/20 0.38
FGFR1 P11362 1/20 0.37
FLT1 P17948 1/20 0.37
KDR P35968 1/20 0.37
FLT3 P36888 3/20 0.37
KMT2A Q03164 2/20 0.37
AR P10275 1/20 0.37
MITF O75030 1/20 0.37
LMNA P02545 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6188924 0.91 LMNA (0.39) ALDH1A1MAPTGAAALOX15KMT2A
SCHEMBL6185751 0.89 AR (0.45) ALDH1A1MAPTNGFRGAAPARP1
SCHEMBL6185980 0.84 LMNA (0.41) ALDH1A1MAPTNGFRGAAPARP1
SCHEMBL6191071 0.82 TUBB1 (0.44) ALDH1A1MAPTGAAPTGS1PTGS2
SCHEMBL28358993 0.78 NGFR (0.46) ALDH1A1MAPTNGFRGAAPARP1
SCHEMBL6184788 0.75 MAOA (0.45) MAPTGAAKMT2ALMNARAB9A
SCHEMBL6631783 0.74 NGFR (0.43) ALDH1A1NGFRGAAPARP1CA12
SCHEMBL6189884 0.74 MAOA (0.48) ALDH1A1GAANPSR1POLB
SCHEMBL6189592 0.74 MAOA (0.51) ALDH1A1GAALMNANPSR1POLB
SCHEMBL6189554 0.73 ALDH1A1 (0.46) ALDH1A1MAPTGAAPARP1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554271-A1 SUBSTITUTED INDOLES AND THEIR USE AS HCV INHIBITORS Rigel Pharmaceuticals, Inc. (US) 2005-07-20 EP disclosed
WO-2004035571-A1 SUBSTITUTED INDOLES AND THEIR USE AS HCV INHIBITORS RIGEL PHARMACEUTICALS, INC. (US) 2004-04-29 WO disclosed