SCHEMBL6202065

SCHEMBL6202065

O=C(CC(c1ccc(F)cc1)c1cnccn1)c1ccc(Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.42
KMT2A Q03164 2/20 0.41
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
EPHX2 P34913 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MGAM O43451 1/20 0.39
GAA P10253 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
TP53 P04637 1/20 0.39
VNN1 O95497 1/20 0.39
SLC6A9 P48067 1/20 0.38
SLC6A5 Q9Y345 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
FFAR2 O15552 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201493 0.84 LMNA (0.46) KMT2ACYP2C9CYP2C19EPHX2MGAM
SCHEMBL6201652 0.77 ALDH1A1 (0.43) POLBKMT2ATP53NPC1RAB9A
SCHEMBL6201073 0.75 CYP19A1 (0.53) POLBKMT2ACYP2C9CYP2C19MGAM
SCHEMBL6202063 0.74 MDM2 (0.46) KMT2ACYP2C9CYP2C19KDM4EVNN1
SCHEMBL2142802 0.71 PDPK1 (0.55) POLBKMT2ACYP2C9CYP2C19TP53
SCHEMBL6204077 0.70 MGAM (0.50) POLBKMT2ACYP2C9CYP2C19MGAM
SCHEMBL10908660 0.67 CYP1A2 (0.50) KMT2ACYP2C9CYP2C19KDM4ENPC1
SCHEMBL10906842 0.67 RAB9A (0.65) KMT2AKDM4ENPC1RAB9A
SCHEMBL10908679 0.67 RAB9A (0.65) KMT2ACYP2C9CYP2C19KDM4ENPC1
SCHEMBL7363506 0.65 TBXAS1 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1549600-A1 KETONES AstraZeneca AB (SE) 2005-07-06 EP disclosed
WO-2004011410-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2004-02-05 WO disclosed