SCHEMBL6210230

SCHEMBL6210230

CC(CCNC(=O)c1ccc(-c2cnco2)cc1)CC(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.40
SMYD3 Q9H7B4 2/20 0.37
LMNA P02545 1/20 0.35
GPR119 Q8TDV5 4/20 0.33
TAOK1 Q7L7X3 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PTAFR P25105 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6213640 0.90 ROCK2 (0.38) ROCK2SMYD3LMNAGPR119TAOK1
SCHEMBL6210763 0.89 ROCK2 (0.36) ROCK2GPR119TAOK1
SCHEMBL6212956 0.88 ROCK2 (0.41) ROCK2LMNAGPR119TAOK1PTAFR
SCHEMBL6215209 0.88 ROCK2 (0.40) ROCK2SMYD3LMNAALDH1A1PTAFR
SCHEMBL6208718 0.88 LMNA (0.42) SMYD3LMNAALDH1A1
SCHEMBL6209450 0.88 CXCR3 (0.43) SMYD3LMNAPTAFR
SCHEMBL6211570 0.88 SLC6A5 (0.38) SMYD3LMNA
SCHEMBL6211038 0.88 CTSK (0.41) SMYD3LMNAALDH1A1
SCHEMBL6210489 0.87 CHRM4 (0.39) SMYD3LMNA
SCHEMBL6211651 0.87 NAMPT (0.38) SMYD3LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP claimed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO claimed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed