SCHEMBL6232343

SCHEMBL6232343

Nc1ccc2nc(CN3CCN(c4ccccc4)CC3)ccc2c1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.48
DRD4 P21917 5/20 0.48
DRD2 P14416 3/20 0.48
DRD3 P35462 3/20 0.48
KDM4E B2RXH2 2/20 0.47
FAAH O00519 2/20 0.47
GRM2 Q14416 1/20 0.44
MAPT P10636 2/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 2/20 0.44
MAPK1 P28482 1/20 0.44
GFER P55789 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
GAA P10253 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2921149 0.82 MAOA (0.48) MCHR1DRD2DRD3KDM4EFAAH
SCHEMBL1352039 0.81 MAPT (0.55) MCHR1KDM4EMAPTGAASMN1; SMN2
SCHEMBL6229471 0.81 LMNA (0.50) MCHR1KDM4EFAAHMAPTLMNA
SCHEMBL2926351 0.81 ALDH1A1 (0.47) MCHR1DRD2DRD3KDM4EFAAH
SCHEMBL5764654 0.80 MCHR1 (0.49) MCHR1DRD4DRD2DRD3KDM4E
SCHEMBL6231291 0.80 ALDH1A1 (0.53) MCHR1ALDH1A1LMNAMAPK1
SCHEMBL10364825 0.76 PLAU (0.41) MCHR1DRD2DRD3KDM4EFAAH
SCHEMBL8319517 0.74 FAAH (0.51) DRD4DRD2DRD3KDM4EFAAH
SCHEMBL8323715 0.74 SLC6A4 (0.54) DRD4DRD2DRD3KDM4EFAAH
SCHEMBL8323587 0.73 HTR1A (0.55) DRD4DRD2DRD3KDM4EFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004092181-A9 HETEROCYCLIC MCHR1 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2005-01-27 WO disclosed