SCHEMBL6232429

SCHEMBL6232429

COc1ccc2oc(C(=O)NC(CC3CC3)C(=O)N3CCC4C3C(=O)CN4S(=O)(=O)c3cccc[n+]3[O-])cc2c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 11/20 0.41
TAS1R1 Q7RTX1 11/20 0.41
CTSL P07711 5/20 0.39
CTSS P25774 5/20 0.39
CTSK P43235 5/20 0.39
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
HTR2A P28223 1/20 0.38
BCAT1 P54687 1/20 0.37
CTSV O60911 1/20 0.36
CTSB P07858 1/20 0.36
ACHE P22303 1/20 0.35
TACR2 P21452 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043929 0.90 CTSV (0.32) TAS1R3TAS1R1CTSLCTSSCTSK
SCHEMBL6210152 0.83 CTSK (0.43) TAS1R3TAS1R1CTSLCTSSCTSK
SCHEMBL6242334 0.83 TAS1R3 (0.46) TAS1R3TAS1R1CTSLCTSSCTSK
SCHEMBL6212161 0.83 CTSK (0.41) TAS1R3TAS1R1CTSLCTSSCTSK
SCHEMBL4042300 0.83 CTSK (0.37) TAS1R3TAS1R1CTSLCTSSCTSK
SCHEMBL4045162 0.82 TAS1R3 (0.34) TAS1R3TAS1R1CTSK
SCHEMBL4043593 0.81 USP2 (0.33) TAS1R3TAS1R1CTSK
SCHEMBL4043294 0.81 CTSS (0.44) CTSLCTSSCTSKCTSV
SCHEMBL4049248 0.80 CTSV (0.31) TAS1R3TAS1R1CTSLCTSSBCAT1
SCHEMBL4040036 0.79 CTSK (0.54) CTSLCTSSCTSKCTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed