SCHEMBL6233705

SCHEMBL6233705

FC(F)(F)c1cccc(Nc2ncco2)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.40
SCN9A Q15858 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
P2RX7 Q99572 11/20 0.36
AURKA O14965 1/20 0.36
DHODH Q02127 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
TRPV1 Q8NER1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6234222 0.80 ULK1 (0.38) SCN9AALDH1A1TDP1AURKADHODH
SCHEMBL6237353 0.71 RAPGEF4 (0.49) ALDH1A1DHODH
SCHEMBL15937997 0.69 KDM4E (0.41) ALDH1A1TDP1
SCHEMBL6237657 0.69 AURKA (0.57) ALDH1A1TDP1AURKADHODH
SCHEMBL6623767 0.68 CCR4 (0.52) ALDH1A1TDP1
SCHEMBL6236093 0.68 CDK4 (0.40) SCN9A
SCHEMBL11404979 0.68 P2RX7 (0.44) NOTUMALDH1A1TDP1P2RX7
SCHEMBL2590517 0.68 P2RX7 (0.49) NOTUMALDH1A1TDP1P2RX7TRPV1
SCHEMBL30041659 0.67 EPHX2 (0.48) SCN9ADHODH
SCHEMBL6240725 0.67 TDO2 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005005382-A2 COMPOUNDS, COMPOSITIONS AND METHODS CYTOKINETICS, INC. (US) 2005-01-20 WO disclosed