SCHEMBL630786

SCHEMBL630786

Cc1ccccc1C[C@@H](N)NC(=O)O[C@H]1CCCCN1S(=O)(=O)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.46
PKM P14618 1/20 0.44
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.41
MMP1 P03956 5/20 0.41
ADAM17 P78536 3/20 0.41
MMP13 P45452 2/20 0.41
FKBP1A P62942 5/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPK1 P28482 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL631739 0.85 TDP1 (0.56) TDP1PKMLMNAPOLBFKBP1A
SCHEMBL630767 0.84 ITGB1 (0.46) TDP1PKMLMNAPOLBFKBP1A
SCHEMBL631469 0.83 ALDH1A1 (0.44) TDP1PKMLMNAPOLBFKBP1A
SCHEMBL631775 0.83 LMNA (0.47) PKMLMNAALDH1A1
SCHEMBL631343 0.83 PKM (0.43) TDP1PKMLMNAPOLBFKBP1A
SCHEMBL630266 0.82 ITGB1 (0.49) TDP1PKMLMNAPOLBALDH1A1
SCHEMBL631194 0.78 ITGB1 (0.47) TDP1PKMLMNAFKBP1AALDH1A1
SCHEMBL13206975 0.76 TDP1 (0.54) TDP1PKMLMNAPOLBFKBP1A
SCHEMBL8268319 0.76 TDP1 (0.54) TDP1PKMLMNAPOLBFKBP1A
SCHEMBL631233 0.76 FKBP1A (0.46) TDP1PKMLMNAPOLBFKBP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778637-B1 FKBP-binding composition and pharmaceutical use thereof AVENTIS PHARMA INC (US) 2012-02-22 EP claimed