Higenamine

Higenamine

SCHEMBL636788

Oc1ccc(CC2NCCc3cc(O)c(O)cc32)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 1.00
DRD4 P21917 2/20 1.00
KDM1A O60341 1/20 1.00
TBXA2R P21731 6/20 0.80
ADRB2 P07550 5/20 0.79
MEN1 O00255 1/20 0.79
ABL1 P00519 1/20 0.79
ALPL P05186 1/20 0.79
GAA P10253 1/20 0.79
KMT2A Q03164 1/20 0.79
RIN1 Q13671 1/20 0.79
KDM4E B2RXH2 1/20 0.74
MAPT P10636 1/20 0.74
PKM P14618 1/20 0.74
ADRB1 P08588 1/20 0.70
BCHE P06276 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(+)-Higenamine SCHEMBL5898913 1.00 DRD2 (1.00) DRD2DRD4KDM1ATBXA2RADRB2
(+)-Higenamine SCHEMBL30464469 1.00 DRD2 (1.00) DRD2DRD4KDM1ATBXA2RADRB2
(-)-Higenamine SCHEMBL29365055 1.00 DRD2 (1.00) DRD2DRD4KDM1ATBXA2RADRB2
(-)-Higenamine SCHEMBL5898911 1.00 DRD2 (1.00) DRD2DRD4KDM1ATBXA2RADRB2
Higenamine SCHEMBL30105922 1.00 DRD2 (1.00) DRD2DRD4KDM1ATBXA2RADRB2
(-)-Higenamine SCHEMBL5898916 0.99 DRD2 (0.97) DRD2DRD4KDM1ATBXA2RADRB2
(-)-Higenamine SCHEMBL29374757 0.99 DRD2 (0.97) DRD2DRD4KDM1ATBXA2RADRB2
(+)-Higenamine SCHEMBL5898932 0.99 DRD2 (0.97) DRD2DRD4KDM1ATBXA2RADRB2
Higenamine SCHEMBL28478764 0.99 DRD2 (0.97) DRD2DRD4KDM1ATBXA2RADRB2
Higenamine SCHEMBL29623874 0.99 DRD2 (0.97) DRD2DRD4KDM1ATBXA2RADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1175 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260125725-A1 Compositions And Methods For Making Benzylisoquinoline Alkaloids, Morphinan Alkaloids, Thebaine, And Derivatives Thereof ANTHEIA INC (US) 2026-05-07 US claimed
US-20260121027-A1 POSITIVE ELECTRODE FOR RECHARGEABLE LITHIUM BATTERY AND RECHARGEABLE LITHIUM BATTERY INCLUDING THE SAME SAMSUNG SDI CO., LTD. (KR) 2026-04-30 US claimed
US-20260110656-A1 ELECTROCHEMICAL SENSOR PREPARED FROM NIOBIUM CARBIDE-REDUCED GRAPHENE OXIDE AEROGEL COMPOSITE MATERIAL AND ITS UTILIZATION NATIONAL TAIPEI UNIVERSITY OF TECHNOLOGY (TW) 2026-04-23 US claimed
EP-4722714-A1 SIMULTANEOUS ANALYSIS OF FOOD-BORNE DOPING SUBSTANCES USING LIQUID CHROMATOGRAPHY-MASS SPECTROMETRY (VFD: VACCINE FOR FOODBORNE DOPING) Korea Institute of Science and Technology (KR) 2026-04-08 EP claimed
US-20260074280-A1 Rechargeable Lithium Batteries SAMSUNG SDI CO LTD (KR) 2026-03-12 US claimed
US-20250388939-A1 RECOMBINANT HOST CELLS WITH IMPROVED PRODUCTION OF L-DOPA, DOPAMINE, S-NOROCLAURINE OR DERIVATIVES THEREOF RIVER STONE BIOTECH APS (DK) 2025-12-25 US claimed
EP-4615963-A1 GENETICALLY MODIFIED BENZYLISOQUINOLINE ALKALOID-PRODUCING HOST CELLS WITH MODIFIED EFFLUX TRANSPORTER GENE EXPRESSION River Stone Biotech ApS (DK) 2025-09-17 EP claimed
EP-4599048-A1 COMPOSITIONS AND METHODS FOR SMALL MOLECULE BASED EXPANSION OF PLURIPOTENT STEM CELLS Trailhead Biosystems Inc. (US) 2025-08-13 EP claimed
US-12371722-B2 Recombinant host cells with improved production of L-DOPA, dopamine, S-noroclaurine or derivatives thereof RIVER STONE BIOTECH APS (DK) 2025-07-29 US claimed
US-20250213647-A1 CHEMOKINE RECEPTORS AND ALPHA1 ADRENERGIC RECEPTORS/VASOPRESSIN RECEPTORS 1A HETEROMERS AS DRUG TARGETS FOR DISEASE UNIVERSITY OF SOUTH FLORIDA 2025-07-03 US claimed
EP-2376073-A2 DERMAL APPLICATION OF VASOCONSTRICTORS Zachar, Oron (IL) 2011-10-19 EP claimed
WO-2011084459-A1 PPAR-SPARING THIAZOLIDINEDIONES AND COMBINATIONS FOR THE TREATMENT OF OBESITY AND OTHER METABOLIC DISEASES METABOLIC SOLUTIONS DEVELOPMENT COMPANY (US) 2011-07-14 WO claimed
WO-2011084456-A1 PPAR-SPARING THIAZOLIDINEDIONES AND COMBINATIONS FOR THE TREATMENT OF DIABETES MELLITUS AND OTHER METABOLIC DISEASES METABOLIC SOLUTIONS DEVELOPMENT COMPANY (US) 2011-07-14 WO claimed
CN-102107006-A Coupling medicament for treating diabetes mellitus and medicinal application thereof CHIFCON DRUG DISCOVERY SUZHOU INC 2011-06-29 CN claimed
WO-2011075514-A1 PPAR-SPARING THIAZOLIDINEDIONES AND COMBINATIONS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES METABOLIC SOLUTIONS DEVELOPMENT COMPANY (US) 2011-06-23 WO claimed
US-20110144209-A1 USE OF VASOCONSTRICTORS ZACHAR ORON 2011-06-16 US claimed
EP-2313037-A1 DERMAL APPLICATION OF VASOCONSTRICTORS Zachar, Oron (IL) 2011-04-27 EP claimed
WO-2010063030-A2 DERMAL APPLICATION OF VASOCONSTRICTORS FEIGELSON, DANIEL (IL) 2010-06-03 WO claimed
WO-2010001391-A1 DERMAL APPLICATION OF VASOCONSTRICTORS ZACHAR ORON (IL) 2010-01-07 WO claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260074280-A1 Rechargeable Lithium Batteries SLC9A2, SLC9A1, CACNA2D1 DRD2 2499/4885DRD4 2396/4885KDM1A 1366/4885
US-20260125725-A1 Compositions And Methods For Making Benzylisoquinoline Alkaloids, Morphinan Alkaloids, Thebaine, And Derivatives Thereof OPRD1, OPRM1, OPRK1 DRD2 218/4885DRD4 374/4885KDM1A 3075/4885
US-20260110656-A1 ELECTROCHEMICAL SENSOR PREPARED FROM NIOBIUM CARBIDE-REDUCED GRAPHENE OXIDE AEROGEL COMPOSITE MATERIAL AND ITS UTILIZATION OGG1, SCO2, CPNE4 DRD2 1615/4885DRD4 1008/4885KDM1A 2977/4885
US-20260121027-A1 POSITIVE ELECTRODE FOR RECHARGEABLE LITHIUM BATTERY AND RECHARGEABLE LITHIUM BATTERY INCLUDING THE SAME CACNA2D4, SLC8A1, SLC9A2 DRD2 2300/4885DRD4 1998/4885KDM1A 2536/4885
US-20250388939-A1 RECOMBINANT HOST CELLS WITH IMPROVED PRODUCTION OF L-DOPA, DOPAMINE, S-NOROCLAURINE OR DERIVATIVES THEREOF DBH, DDT, COMT DRD2 989/4885DRD4 1463/4885KDM1A 2519/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.