Telmesteine

Telmesteine

SCHEMBL637246

CCOC(=O)N1CSC[C@H]1C(=O)O

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.53
PREP P48147 2/20 0.43
RAB9A P51151 1/20 0.39
TSHR P16473 1/20 0.36
PPM1B O75688 1/20 0.36
PTPN1 P18031 1/20 0.36
PPP1CC P36873 1/20 0.36
ATM Q13315 1/20 0.34
RECQL P46063 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Telmesteine SCHEMBL1425417 1.00 ACE (0.53) ACEPREPRAB9ATSHRPPM1B
SCHEMBL6706811 0.86 ACE (0.47) ACEPREPRAB9ATSHRATM
SCHEMBL7769271 0.85 PREP (0.40) ACEPREPTSHRATMRECQL
SCHEMBL7769272 0.85 GAA (0.42) ACEPREPTSHRGAA
Telmesteine SCHEMBL7269300 0.81 GSR (0.46) ACEPREP
Telmesteine SCHEMBL7269301 0.81 GSR (0.46) ACEPREP
SCHEMBL5494135 0.80 ACE (0.54) ACEPREPRAB9AATM
SCHEMBL19084116 0.79 ACE (0.55) ACEPREPTSHR
SCHEMBL6051964 0.79 ACE (0.55) ACEPREPTSHR
SCHEMBL202300 0.78 ACE (0.48) ACEPREPATMRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 418 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260130899-A1 METHOD OF TREATMENT FOR PREVENTION OF GLUCOCORTICOID TOXICITY AND/OR ENHANCEMENT OF MUSCLE REGENERATION VIA NEUTROPHIL ELASTASE INHIBITION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2026-05-14 US claimed
US-20240216353-A1 METHOD OF TREATMENT FOR PREVENTION OF GLUCOCORTICOID TOXICITY AND/OR ENHANCEMENT OF MUSCLE REGENERATION VIA NEUTROPHIL ELASTASE INHIBITION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2024-07-04 US claimed
US-20210315873-A1 METHOD OF TREATMENT FOR PREVENTION OF GLUCOCORTICOID TOXICITY AND/OR ENHANCEMENT OF MUSCLE REGENERATION VIA NEUTROPHIL ELASTASE INHIBITION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2021-10-14 US claimed
CN-109248319-A Contain the pharmaceutical composition for taking charge of smooth class compound and aspirin 郜建敏 2019-01-22 CN claimed
CN-107157976-A Application of the compound of thioether acids structure in medicament for resisting platelet aggregation is prepared 北京北朋科技有限公司 2017-09-15 CN claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20140178399-A1 ROLE OF ADAM10 AND ITS RELEVANCE TO DISEASE AND THERAPEUTICS UNIVERSITY OF CHICAGO (US) 2014-06-26 US claimed
EP-2637679-A1 ROLE OF ADAM10 AND ITS RELEVANCE TO DISEASE AND THERAPEUTICS The University of Chicago (US) 2013-09-18 EP claimed
US-8431601-B2 Topical compositions comprising telmesteine for treating dermatological disorders SINCLAIR PHARMACEUTICALS LTD. (GB) 2013-04-30 US claimed
US-8268352-B2 Modified release composition for highly soluble drugs TORRENT PHARMACEUTICALS LIMITED (IN) 2012-09-18 US claimed
US-20060247183-A1 Compositions and methods for the treatment of inflammatory conditions of mucosae, skin and the eye SINCLAIR PHARMACEUTICALS LTD. (GB) 2006-11-02 US claimed
EP-1670464-A1 TOPICAL COMPOSITIONS COMPRISING TELMESTEINE FOR TREATING DERMATOLOGICAL DISORDERS Sinclair Pharmaceuticals Limited (GB) 2006-06-21 EP claimed
US-20060024365-A1 Novel dosage form VAYA NAVIN 2006-02-02 US claimed
US-20060018933-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20060018934-A1 Novel drug delivery system TORRENT PHARMACEUTICALS LIMITED (IN) 2006-01-26 US claimed
US-20050143324-A1 Compositions and methods for the treatment of inflammatory conditions of mucosae, skin and the eye SINCLAIR PHARMACEUTICALS, LTD. 2005-06-30 US claimed
WO-2005037275-A1 TOPICAL COMPOSITIONS COMPRISING TELMESTEINE FOR TREATING DERMATOLOGICAL DISORDERS SINCLAIR PHARMACEUTICALS LIMITED (GB) 2005-04-28 WO claimed
EP-1494692-A1 TOPICAL PHARMACEUTICAL COMPOSITIONS COMPRISING PROANTHOCYANIDINS FOR THE TREATMENT OF DERMATITIS Sinclair Pharmaceuticals Limited (GB) 2005-01-12 EP claimed
WO-2003084553-A1 TOPICAL PHARMACEUTICAL COMPOSITIONS COMPRISING PROANTHOCYANIDINS FOR THE TREATMENT OF DERMATITIS SINCLAIR PHARMACEUTICALS LIMITED (GB) 2003-10-16 WO claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260130899-A1 METHOD OF TREATMENT FOR PREVENTION OF GLUCOCORTICOID TOXICITY AND/OR ENHANCEMENT OF MUSCLE REGENERATION VIA NEUTROPHIL ELASTASE INHIBITION SERPINB1, ELANE, CELA1 ACE 151/4885PREP 269/4885RAB9A 2398/4885
US-20140178399-A1 ROLE OF ADAM10 AND ITS RELEVANCE TO DISEASE AND THERAPEUTICS ADAM10, ADAM8, ADAM17 ACE 93/4885PREP 41/4885RAB9A 787/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.