SCHEMBL644137

SCHEMBL644137

Oc1cccc(O)c1SS

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.45
ALOX15 P16050 5/20 0.45
HPGD P15428 5/20 0.45
HSD17B10 Q99714 5/20 0.45
CA2 P00918 3/20 0.45
RECQL P46063 3/20 0.45
TDP1 Q9NUW8 3/20 0.45
LMNA P02545 3/20 0.45
EGFR P00533 2/20 0.45
FYN P06241 2/20 0.45
MMP9 P14780 2/20 0.45
CA1 P00915 2/20 0.45
ADAMTS4 O75173 1/20 0.45
MMP2 P08253 1/20 0.45
MMP8 P22894 1/20 0.45
CA6 P23280 1/20 0.45
CDK2 P24941 1/20 0.45
MMP12 P39900 1/20 0.45
ADAMTS5 Q9UNA0 1/20 0.45
MAPT P10636 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8888927 0.75 ALDH1A1 (0.50) ALDH1A1ALOX15HPGDHSD17B10CA2
SCHEMBL9853388 0.71 ALDH1A1 (0.45) ALDH1A1ALOX15HPGDHSD17B10CA2
SCHEMBL3917019 0.71 ALOX15 (0.45) ALDH1A1ALOX15HPGDHSD17B10CA2
SCHEMBL7513765 0.70 ALOX15 (0.52) ALDH1A1ALOX15HPGDHSD17B10CA2
SCHEMBL6274433 0.69 USP2 (0.70) ALDH1A1HPGDHSD17B10RECQLTDP1
SCHEMBL5179392 0.69
SCHEMBL24718435 0.65 ALDH1A1 (0.39) ALDH1A1ALOX15HPGDHSD17B10CA2
SCHEMBL10887948 0.65 TSHR (0.54) ALDH1A1ALOX15HPGDHSD17B10CA2
SCHEMBL2865709 0.65 ALDH1A1 (0.43) ALDH1A1ALOX15HPGDHSD17B10CA2
SCHEMBL1358980 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119103-B2 Bifunctional resorcinol, thioresorcinol, and dithioresorcinol derivative metal chelating conjugates MALLINCKRODT LLC (US) 2012-02-21 US disclosed
US-20100055043-A1 Poly-Halo Metal X-ray Contrast Agents MALLINCKRODT INC. 2010-03-04 US disclosed
EP-2089063-A2 X-RAY CONTRAST AGENTS COMPRISING A METAL CHELATE AND A POLYHALOGENATED PHENOL, THIOPHENOL, RESORCINOL, THIORESORCINOL OR DITHIORESORCINOL Mallinckrodt Inc. (US) 2009-08-19 EP disclosed
US-20090082324-A1 Bifunctional Resorcinol, Thioresorcinol, and Dithioresorcinol Derivative Metal Chelating Conjugates INFACARE PHARMACEUTICAL CORPORATION 2009-03-26 US disclosed
EP-1988925-A2 BIFUNCTIONAL RESORCINOL, THIORESORCINOL, AND DITHIORESORCINOL DERIVATIVE METAL CHELATING CONJUGATES MALLINCKRODT, INC. (US) 2008-11-12 EP disclosed
WO-2008060399-A2 X-RAY CONTRAST AGENTS COMPRISING A METAL CHELATE AND A POLYHALOGENATED PHENOL, THIOPHENOL, RESORCINOL, THIORESORCINOL OR DITHIORESORCINOL MALLINCKRODT INC. (US) 2008-05-22 WO disclosed
WO-2007100563-A2 BIFUNCTIONAL RESORCINOL, THIORESORCINOL, AND DITHIORESORCINOL DERIVATIVE METAL CHELATING CONJUGATES MALLINCKRODT INC. (US) 2007-09-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090082324-A1 Bifunctional Resorcinol, Thioresorcinol, and Dithioresorcinol Derivative Metal Chelating Conjugates SPR, QDPR, SLC40A1 ALDH1A1 716/4885ALOX15 4499/4885HPGD 2378/4885
US-20100055043-A1 Poly-Halo Metal X-ray Contrast Agents SLC39A3, ZNF277, TPR ALDH1A1 3268/4885ALOX15 4178/4885HPGD 2704/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.