SCHEMBL6446578

SCHEMBL6446578

N#CCCNC(=O)C(CNC(=O)c1cccc(CCl)c1)c1ccc2ccccc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.41
GUSB P08236 1/20 0.40
CTSK P43235 6/20 0.37
CTSL P07711 5/20 0.37
CTSS P25774 5/20 0.37
OPRM1 P35372 1/20 0.36
TMEM97 Q5BJF2 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
HDAC3 O15379 4/20 0.36
HDAC4 P56524 4/20 0.36
HDAC1 Q13547 4/20 0.36
HDAC7 Q8WUI4 4/20 0.36
HDAC2 Q92769 4/20 0.36
HDAC10 Q969S8 4/20 0.36
HDAC11 Q96DB2 4/20 0.36
HDAC8 Q9BY41 4/20 0.36
HDAC6 Q9UBN7 4/20 0.36
HDAC9 Q9UKV0 4/20 0.36
HDAC5 Q9UQL6 4/20 0.36
CTSB P07858 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6447466 0.90 CTSL (0.47) ATMCTSKCTSLCTSSCTSB
SCHEMBL6446797 0.90 CTSS (0.43) ATMGUSBCTSKCTSLCTSS
SCHEMBL6446599 0.89 GUSB (0.43) GUSBCTSKCTSLCTSSHDAC3
SCHEMBL6447322 0.88 CTSK (0.42) ATMGUSBCTSKCTSLCTSS
SCHEMBL6445190 0.87 GUSB (0.40) GUSBCTSKCTSLCTSSCTSB
SCHEMBL6444201 0.84 CTSL (0.47) ATMCTSLPIN1
SCHEMBL6446493 0.81 CTSL (0.53) ATMCTSKCTSLCTSSHDAC1
SCHEMBL6447506 0.80 CTSL (0.53) CTSKCTSLCTSSCTSBCTSV
SCHEMBL6446969 0.79 KDM4E (0.44) ATMCTSKCTSLCTSSCTSB
SCHEMBL6019767 0.79 CTSL (0.60) CTSKCTSLCTSSCTSBCTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed