SCHEMBL6445190

SCHEMBL6445190

N#CCCNC(=O)C(CNC(=O)c1cccc(CCl)c1)c1ccc(O)cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GUSB P08236 1/20 0.40
CTSL P07711 10/20 0.37
CTSS P25774 6/20 0.36
CTSK P43235 6/20 0.36
CTSV O60911 3/20 0.36
CTSB P07858 3/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GLI1 P08151 1/20 0.35
GLI2 P10070 1/20 0.35
SFN P31947 1/20 0.34
KDM4A O75164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446599 0.92 GUSB (0.43) GUSBCTSLCTSSCTSKCTSV
SCHEMBL6822562 0.90 CTSK (0.47) CTSLCTSSCTSKCTSVCTSB
SCHEMBL6443632 0.88 SFN (0.42) GUSBCTSLCTSSCTSKGAA
SCHEMBL6446578 0.87 ATM (0.41) GUSBCTSLCTSSCTSKCTSV
SCHEMBL6443745 0.85 CTSS (0.47) GUSBCTSLCTSSCTSKCTSB
SCHEMBL6442129 0.83 CTSL (0.49) CTSL
SCHEMBL6447506 0.82 CTSL (0.53) CTSLCTSSCTSKCTSVCTSB
SCHEMBL6446816 0.81 GAA (0.40) GUSBCTSLCTSSCTSKCTSV
SCHEMBL6442019 0.80 CTSS (0.42) GUSBCTSLCTSSCTSKCTSB
SCHEMBL6020870 0.80 CTSL (0.61) CTSLCTSSCTSKCTSVCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed