SCHEMBL646260

SCHEMBL646260

C=CC(O)Nc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.44
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
TGM2 P21980 1/20 0.42
ALDH1A1 P00352 7/20 0.39
TSHR P16473 6/20 0.39
HSD17B10 Q99714 5/20 0.39
ALOX15 P16050 3/20 0.39
ALOX12 P18054 3/20 0.39
CYP3A4 P08684 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
LMNA P02545 1/20 0.39
THRB P10828 1/20 0.39
RECQL P46063 1/20 0.39
ATM Q13315 1/20 0.39
IDO1 P14902 1/20 0.39
CTSD P07339 1/20 0.36
CYP1A2 P05177 1/20 0.35
MAPK1 P28482 2/20 0.35
PTGS1 P23219 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21787328 0.78 TDP1 (0.46) TDP1CA9ALDH1A1TSHRHSD17B10
SCHEMBL6255896 0.78 MAPT (0.39) TDP1CA12CA9ALDH1A1HSD17B10
SCHEMBL3952756 0.78 CA1 (0.46) TDP1CA12TGM2ALDH1A1CYP3A4
SCHEMBL4632504 0.78 ALDH1A1 (0.46) TDP1ALDH1A1HSD17B10ALOX15ALOX12
SCHEMBL21891545 0.77 CA12 (0.47) TDP1CA12CA9TGM2ALDH1A1
SCHEMBL22225161 0.77 MMP2 (0.31) CA12CA9TGM2
SCHEMBL10987834 0.75 TYR (0.41) ALDH1A1HSD17B10PTGS2
SCHEMBL2898716 0.75
SCHEMBL28296933 0.74 TDP1 (0.46) TDP1CA12CA9ALDH1A1TSHR
SCHEMBL27269638 0.73 TDP1 (0.50) TDP1CA12CA9TGM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 116 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1414803-B1 PYRAZOLYLCARBOXANILIDES AS FUNGICIDES BAYER CROPSCIENCE AG (DE) 2012-12-12 EP claimed
US-20040204470-A1 Pyrazoylcarboxanilides as fungicides BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2004-10-14 US claimed
US-4235730-A DISPERSANTS TEXACO INC. (US) 1980-11-25 US claimed
JP-56106600-A None JP disclosed
US-20240109862-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH PFIZER INC. 2024-04-04 US disclosed
WO-2021095091-A1 AMINOARYL DERIVATIVE, INTERMEDIATE OF SAME, METHOD FOR PRODUCING SAID AMINOARYL DERIVATIVE, AND METHOD FOR PRODUCING SAID INTERMEDIATE 藤本化学製品株式会社 2021-05-20 WO disclosed
US-10450297-B2 Sulfonyl amide derivatives for the treatment of abnormal cell growth PFIZER, INC. (US) 2019-10-22 US disclosed
US-20190047979-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH PFIZER (US) 2019-02-14 US disclosed
EP-1566693-B1 Use of a Resist Composition for Immersion Exposure and Pattern Formation Method Using the Composition FUJIFILM CORP (JP) 2018-05-23 EP disclosed
US-20170327485-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH PFIZER (US) 2017-11-16 US disclosed
US-9777202-B2 Curable composition suitable for the bonding of plasticized PVC SIKA TECHNOLOGY AG (CH) 2017-10-03 US disclosed
WO-1997027236-A1 POLY(OXYPROPYLENE/OXYETHYLENE) RANDOM POLYOLS USEFUL IN PREPARING FLEXIBLE HIGH RESILIENCE FOAM WITH REDUCED TENDENCIES TOWARD SHRINKAGE AND FOAM PREPARED THEREWITH ARCO CHEMICAL TECHNOLOGY, L.P. (US) 1997-07-31 WO disclosed
EP-0273390-B1 Radiation curable resin composition for use in magnetic recording media MITSUBISHI RAYON CO (JP) 1996-08-14 EP disclosed
US-4963639-A (METH)ACRYLATED POLYURETHANE MITSUBISHI RAYON COMPANY, LTD. (JP) 1990-10-16 US disclosed
US-4672071-A Antihypertensive dihydropyridine compositions, optical isomers and intermediates SYNTEX (U.S.A.) INC. (US) 1987-06-09 US disclosed
EP-0191448-A2 Antihypertensive dihydropyridine derivatives SYNTEX (U.S.A.) INC. (US) 1986-08-20 EP disclosed
US-4595690-A Hypotensive agents SYNTEX (U.S.A.) INC. (US) 1986-06-17 US disclosed
JP-S56106600-A NOVEL DETERMINING METHOD OF HYDROGEN PEROXIDE WAKO PURE CHEM IND LTD 1981-08-24 JP disclosed
US-4009201-A PARTIALLY OR FULLY QUATERNIZED POLYAMINE ESTERS OF ACRYLIC ACIDS ALCOLAC INC. (US) 1977-02-22 US disclosed
US-3955984-A STYRYL DYES FUJI PHOTO FILM CO., LTD. (JA) 1976-05-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10450297-B2 Sulfonyl amide derivatives for the treatment of abnormal cell growth GPR119, INSR, LYAR TDP1 4027/4885CA12 4011/4885CA9 2755/4885
US-20040204470-A1 Pyrazoylcarboxanilides as fungicides CYP1A1, CYP1B1, CYP2E1 TDP1 864/4885CA12 3043/4885CA9 1775/4885
US-20170327485-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH GPR119, INSR, LYAR TDP1 4027/4885CA12 4011/4885CA9 2755/4885
US-20190047979-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH GPR119, INSR, LYAR TDP1 4027/4885CA12 4011/4885CA9 2755/4885
US-20240109862-A1 SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH GPR119, INSR, LYAR TDP1 4027/4885CA12 4011/4885CA9 2755/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.