SCHEMBL6467902

SCHEMBL6467902

CC(C)CC(NC(=O)O)C(=O)NC(CCc1ccccc1)C(=O)c1nc(C(=O)N2CCc3ccccc3C2)co1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB2 P49721 3/20 0.44
PSMB1 P20618 2/20 0.44
CTSS P25774 5/20 0.41
CTSB P07858 5/20 0.41
CTSK P43235 4/20 0.41
CTSL P07711 3/20 0.41
MMP1 P03956 1/20 0.41
MMP3 P08254 1/20 0.41
MMP9 P14780 1/20 0.41
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
PSMB5 P28074 6/20 0.39
PSMB8 P28062 2/20 0.39
PSMB10 P40306 2/20 0.39
HTT P42858 1/20 0.39
TMPRSS11D O60235 1/20 0.39
CTRL P40313 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6466880 0.85 PSMB2 (0.45) PSMB2PSMB1CTSSCTSBCTSK
SCHEMBL6465946 0.85 ALDH1A1 (0.41) PSMB2PSMB1CTSSCTSBCTSK
SCHEMBL7045294 0.80 CTSL (0.52) CTSSCTSBCTSKCTSL
SCHEMBL6466271 0.80 MMP9 (0.44) CTSSCTSBCTSKCTSLMMP1
SCHEMBL6464783 0.80 MMP9 (0.44) CTSSCTSBCTSKCTSLMMP1
SCHEMBL6466269 0.80 MMP9 (0.44) CTSSCTSBCTSKCTSLMMP1
SCHEMBL6464784 0.80 ANPEP (0.48) CTSSCTSBCTSKCTSLMMP3
SCHEMBL7042164 0.80 CTSL (0.46) CTSSCTSBCTSKCTSL
SCHEMBL6063745 0.79 CTSL (0.54) CTSSCTSBCTSKCTSL
SCHEMBL6477967 0.78 MMP3 (0.44) CTSSCTSBCTSKCTSLMMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed