SCHEMBL6468626

SCHEMBL6468626

NC(=O)C(CC1CCCCC1)C(CCc1ccccc1)C(=O)c1nc2ccccc2o1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSS P25774 7/20 0.44
FAAH O00519 2/20 0.43
CES1 P23141 1/20 0.43
DAGLA Q9Y4D2 1/20 0.43
XDH P47989 3/20 0.42
MMP1 P03956 1/20 0.41
MMP2 P08253 1/20 0.41
MMP3 P08254 1/20 0.41
PRSS8 Q16651 2/20 0.39
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
CTSK P43235 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CCR1 P32246 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6463414 1.00 CTSS (0.44) CTSSFAAHCES1DAGLAXDH
SCHEMBL6463782 0.87 CTSS (0.43) CTSSFAAHCES1DAGLAXDH
SCHEMBL6467110 0.86 CTSS (0.44) CTSSFAAHCES1CTSKNPC1
SCHEMBL6466904 0.84 DAGLA (0.50) FAAHCES1DAGLAXDHPRSS8
SCHEMBL6467344 0.83 PRSS8 (0.45) CTSSFAAHCES1DAGLAMMP1
SCHEMBL6473317 0.81 MMP1 (0.40) CTSSFAAHCES1DAGLAXDH
SCHEMBL6465885 0.81 XDH (0.47) CTSSFAAHCES1DAGLAXDH
SCHEMBL6472179 0.80 MMP3 (0.44) CTSSFAAHCES1MMP1MMP2
SCHEMBL5671486 0.80 CTSS (0.39) CTSSFAAHCES1DAGLAXDH
SCHEMBL6467360 0.79 CNR1 (0.49) MMP1MMP2MMP3NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed