SCHEMBL6526664

SCHEMBL6526664

CC(C)(C)OC(=O)NCc1cccc(CC(=O)N[C@](C)(CN2CCCC2)c2ccccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GLS O94925 11/20 0.49
ROCK2 O75116 1/20 0.42
CYP2D6 P10635 1/20 0.41
OPRK1 P41145 1/20 0.41
NPFFR1 Q9GZQ6 1/20 0.41
NPFFR2 Q9Y5X5 1/20 0.41
SIGMAR1 Q99720 2/20 0.40
BRD4 O60885 2/20 0.40
NAMPT P43490 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6526565 0.86 KCNA5 (0.40) GLSCYP2D6OPRK1NPFFR1NPFFR2
SCHEMBL13293669 0.77 ROCK2 (0.55) GLSROCK2CYP2D6NPFFR1NPFFR2
SCHEMBL28211519 0.74 GLS (0.62) GLSBRD4
SCHEMBL2787151 0.74 GLS (0.58) GLSBRD4NAMPT
SCHEMBL5843322 0.73 OPRK1 (0.77) CYP2D6OPRK1
SCHEMBL185365 0.72 ATM (0.55) GLSBRD4NAMPT
SCHEMBL14367982 0.72 PRMT6 (0.56) GLSROCK2BRD4NAMPT
SCHEMBL14986954 0.71 GLS (0.57) GLSBRD4NAMPT
SCHEMBL8786913 0.71 GLS (0.57) GLSBRD4NAMPT
SCHEMBL2066840 0.71 SIGMAR1 (0.46) CYP2D6NPFFR1NPFFR2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005004796-A2 SULFONYLAMINO PHENYLACETAMIDE DERIVATIVES AND METHODS OF THEIR USE ADOLOR CORPORATION (US) 2005-01-20 WO disclosed