SCHEMBL653867

SCHEMBL653867

O=C(NC12CC3CC(CC(C3)C1)C2)N[C@H]1CC[C@H](Oc2ccc(C(=O)O)cc2)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 20/20 1.00
CYP2C19 P33261 1/20 0.64
EPHX1 P07099 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14150188 1.00 EPHX2 (1.00) EPHX2CYP2C19EPHX1
SCHEMBL18465002 1.00 EPHX2 (1.00) EPHX2CYP2C19EPHX1
SCHEMBL653866 1.00 EPHX2 (1.00) EPHX2CYP2C19EPHX1
SCHEMBL12931839 0.89 EPHX2 (0.80) EPHX2
SCHEMBL15272724 0.88 EPHX2 (1.00) EPHX2
SCHEMBL15272793 0.88 EPHX2 (1.00) EPHX2
SCHEMBL1062800 0.87 EPHX2 (1.00) EPHX2
SCHEMBL3195594 0.87 EPHX2 (1.00) EPHX2
SCHEMBL1065991 0.87 EPHX2 (1.00) EPHX2
SCHEMBL3183514 0.87 EPHX2 (1.00) EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 84 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260130877-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS THE REGENTS OF THE UNIV OF CALIFORNIA (US) 2026-05-14 US claimed
US-20230301949-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS CHIBA UNIVERSITY (JP) 2023-09-28 US claimed
US-11723929-B2 Methods of improving cell-based therapy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-08-15 US claimed
US-11690837-B2 Methods of improving cell-based therapy THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-07-04 US claimed
US-11564914-B2 Methods of treating bone loss THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-01-31 US claimed
US-20220202744-A1 METHODS OF TREATING MENTAL DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2022-06-30 US claimed
US-20210378995-A1 METHODS AND TOPICAL PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF SKIN MICROVASCULAR DYSFUNCTION UNIVERSITE DE ROUEN NORMANDIE (FR) 2021-12-09 US claimed
EP-3863639-A1 METHODS AND TOPICAL PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF SKIN MICROVASCULAR DYSFUNCTION INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2021-08-18 EP claimed
US-20210145891-A1 METHODS OF IMPROVING CELL-BASED THERAPY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2021-05-20 US claimed
US-20200306232-A1 METHODS OF TREATING BONE LOSS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2020-10-01 US claimed
US-20190125696-A1 METHODS OF TREATING MENTAL DISORDERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-05-02 US claimed
WO-2018231702-A1 METHODS OF IMPROVING CELL-BASED THERAPY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-12-20 WO claimed
US-20180200244-A1 METHODS OF IMPROVING CELL-BASED THERAPY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-07-19 US claimed
US-20180185309-A1 METHODS AND COMPOSITIONS FOR TREATING NEPHROPATHY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2018-07-05 US claimed
US-7662910-B2 Inhibitors for the soluble epoxide hydrolase THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2010-02-16 US claimed
US-20260130877-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS THE REGENTS OF THE UNIV OF CALIFORNIA (US) 2026-05-14 US disclosed
US-12485107-B2 Methods for the prevention or treatment of cytokine storm BETH ISRAEL DEACONESS MEDICAL CENTER, INC. (US) 2025-12-02 US disclosed
US-7662910-B2 Inhibitors for the soluble epoxide hydrolase THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2010-02-16 US disclosed
WO-2009062073-A1 ALLEVIATING NEUROPATHIC PAIN WITH EETS AND SEH INHIBITORS REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2009-05-14 WO disclosed
WO-2009020960-A1 PREPARATION OF NOVEL 1,3-SUBSTITUTED UREAS AS INHIBITORS OF SOLUBLE EPOXIDE HYDROLASE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2009-02-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200306232-A1 METHODS OF TREATING BONE LOSS EPHX1, NCEH1, SOST EPHX2 4/4885CYP2C19 3862/4885EPHX1 1/4885
US-20230301949-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS FABP7, ADH1B, ELOVL1 EPHX2 51/4885CYP2C19 3526/4885EPHX1 25/4885
US-11723929-B2 Methods of improving cell-based therapy EPHX1, EPHX2, NCEH1 EPHX2 2/4885CYP2C19 2261/4885EPHX1 1/4885
US-20180200244-A1 METHODS OF IMPROVING CELL-BASED THERAPY ELOVL1, ELOVL3, IL2 EPHX2 127/4885CYP2C19 3558/4885EPHX1 116/4885
US-20220202744-A1 METHODS OF TREATING MENTAL DISORDERS FAAH, EPHX1, FAAH2 EPHX2 4/4885CYP2C19 799/4885EPHX1 2/4885
US-20260130877-A1 TREATMENT OF NEURODEVELOPMENTAL DISORDERS EED, ICOS, FABP7 EPHX2 10/4885CYP2C19 676/4885EPHX1 8/4885
US-11690837-B2 Methods of improving cell-based therapy ELOVL1, ELOVL3, IL2 EPHX2 127/4885CYP2C19 3558/4885EPHX1 116/4885
US-11564914-B2 Methods of treating bone loss EPHX1, NCEH1, SOST EPHX2 4/4885CYP2C19 3862/4885EPHX1 1/4885
US-12485107-B2 Methods for the prevention or treatment of cytokine storm TNF, PTGES2, IL2 EPHX2 13/4885CYP2C19 2444/4885EPHX1 5/4885
US-20180185309-A1 METHODS AND COMPOSITIONS FOR TREATING NEPHROPATHY GLS, REN, SLC5A2 EPHX2 3353/4885CYP2C19 4879/4885EPHX1 2595/4885
US-20210145891-A1 METHODS OF IMPROVING CELL-BASED THERAPY EPHX1, EPHX2, NCEH1 EPHX2 2/4885CYP2C19 2261/4885EPHX1 1/4885
US-20190125696-A1 METHODS OF TREATING MENTAL DISORDERS FAAH, EPHX1, FAAH2 EPHX2 4/4885CYP2C19 799/4885EPHX1 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.