SCHEMBL6557412

SCHEMBL6557412

CCOc1cccc(OCc2nc3ccccc3c(=O)n2-c2ccc(OC)cc2)c1OC(=O)CC

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 10/20 0.57
MEN1 O00255 1/20 0.56
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
CYP2C19 P33261 1/20 0.56
KMT2A Q03164 1/20 0.56
ALDH1A1 P00352 1/20 0.54
HTR7 P34969 5/20 0.54
USP2 O75604 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6557887 0.93 HTR7 (0.51) PDE10AMEN1KMT2AALDH1A1HTR7
SCHEMBL6555790 0.91 MEN1 (0.52) PDE10AMEN1CYP1A2CYP3A4CYP2D6
SCHEMBL6557990 0.84 ACHE (0.45) PDE10AHTR7
SCHEMBL6555842 0.83 TSHR (0.52) ALDH1A1HTR7USP2
SCHEMBL6557988 0.81 L3MBTL1 (0.51) KMT2AALDH1A1USP2
SCHEMBL6555584 0.80 PDE4A (0.50) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL6557586 0.78 KDM4E (0.52) PDE10AALDH1A1USP2
SCHEMBL6557322 0.77 KDM4E (0.52) PDE10AKMT2AALDH1A1USP2
SCHEMBL6556016 0.77 L3MBTL1 (0.51) PDE10AALDH1A1USP2
SCHEMBL6557964 0.76 ACKR3 (0.52) ALDH1A1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1073643-B1 NEW HETEROCYCLIC COMPOUNDS AND THEIR USE IN MEDICINE, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM REDDYS LAB LTD DR (IN) 2004-12-29 EP disclosed
EP-1073643-A2 NEW HETEROCYCLIC COMPOUNDS AND THEIR USE IN MEDICINE, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 2001-02-07 EP disclosed
WO-1999008501-A2 NEW HETEROCYCLIC COMPOUNDS AND THEIR USE IN MEDICINE, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S RESEARCH FOUNDATION (IN) 1999-02-25 WO disclosed