SCHEMBL6561914

SCHEMBL6561914

N=C(N)c1ccc(NCC#Cc2ccc(C(=O)c3ccccc3)cn2)cc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.43
VNN1 O95497 3/20 0.42
KLK1 P06870 1/20 0.42
KLK5 Q9Y337 1/20 0.42
DHFR P00374 1/20 0.41
MRGPRX1 Q96LB2 1/20 0.38
PRSS1 P07477 4/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
F2 P00734 2/20 0.37
PRSS2 P07478 2/20 0.37
PRSS3 P35030 2/20 0.37
TMPRSS6 Q8IU80 2/20 0.37
ST14 Q9Y5Y6 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7677085 0.84 VNN1 (0.46) GRM5VNN1
SCHEMBL6563625 0.83 PRSS1 (0.43) MRGPRX1PRSS1ALDH1A1HPGDRAB9A
SCHEMBL6563729 0.81 PPARG (0.41) GRM5VNN1DHFR
SCHEMBL7676492 0.79 CCNA2 (0.41) VNN1MRGPRX1PRSS1ALDH1A1RAB9A
SCHEMBL7678092 0.78 F2 (0.40) KLK1KLK5MRGPRX1PRSS1ALDH1A1
SCHEMBL7669697 0.78 MAPK13 (0.40) PRSS1ALDH1A1HPGDRAB9AF2
SCHEMBL7673754 0.76 NQO2 (0.41) MRGPRX1PRSS1ALDH1A1HPGDF2
SCHEMBL6563277 0.75 F2 (0.41) KLK1KLK5MRGPRX1PRSS1F2
SCHEMBL7670696 0.75 KMT2A (0.44) KLK1KLK5MRGPRX1PRSS1RAB9A
SCHEMBL6565262 0.74 ALDH1A1 (0.45) PRSS1ALDH1A1HPGDRAB9AF2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed