SCHEMBL6565262

SCHEMBL6565262

CC(=O)Nc1cc(C(=O)c2ccccc2)ccc1C#CCNc1ccc(C(=N)N)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
POLB P06746 1/20 0.41
HPGD P15428 2/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RAB9A P51151 1/20 0.38
F7 P08709 4/20 0.37
F2 P00734 3/20 0.37
F10 P00742 1/20 0.37
CACNA1B Q00975 1/20 0.36
APBA1 Q02410 1/20 0.36
PLAU P00749 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36
TMPRSS6 Q8IU80 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7669697 0.85 MAPK13 (0.40) ALDH1A1L3MBTL1HPGDRAB9AF2
SCHEMBL7678092 0.85 F2 (0.40) ALDH1A1L3MBTL1HPGDRAB9AF7
SCHEMBL6563625 0.80 PRSS1 (0.43) ALDH1A1L3MBTL1HPGDRAB9AF7
SCHEMBL6561921 0.76 MAPK13 (0.45) ALDH1A1L3MBTL1HPGDMAPTHTT
SCHEMBL6561914 0.74 GRM5 (0.43) ALDH1A1HPGDRAB9AF2PRSS1
SCHEMBL6563277 0.74 F2 (0.41) F7F2F10PLAUPRSS1
SCHEMBL7675043 0.74 F7 (0.42) F7F2F10PLAUPRSS1
SCHEMBL7673754 0.73 NQO2 (0.41) ALDH1A1HPGDMAPTCYP2C9CYP2C19
SCHEMBL6565690 0.71 PLAU (0.54) HTTRAB9AF2F10PLAU
SCHEMBL6565256 0.71 AKR1C3 (0.44) ALDH1A1F7F2F10PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed