SCHEMBL6563563

SCHEMBL6563563

COC(=O)CCN(c1cc(C)c(C#CCNc2ccc(C(=N)N)cc2)cc1C)S(=O)(=O)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
PLAU P00749 2/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
MAPT P10636 6/20 0.36
MMP1 P03956 4/20 0.35
MMP13 P45452 4/20 0.35
MMP9 P14780 3/20 0.35
LMNA P02545 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
F2 P00734 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MMP12 P39900 1/20 0.34
F10 P00742 1/20 0.34
PRSS1 P07477 1/20 0.34
HPN P05981 2/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563500 0.93 PLAU (0.40) SMN1; SMN2ALDH1A1HPGDHTTPLAU
SCHEMBL6563704 0.86 KEAP1 (0.34) SMN1; SMN2ALDH1A1HPGDHTTKEAP1
SCHEMBL6563152 0.84 F2 (0.43) ALDH1A1L3MBTL1F2F10PRSS1
SCHEMBL6565357 0.83 F2 (0.37) ALDH1A1L3MBTL1F2
SCHEMBL6563095 0.82 ALDH1A1 (0.38) SMN1; SMN2ALDH1A1HPGDHTTPLAU
SCHEMBL6563711 0.82 ADAM17 (0.47) KEAP1NFE2L2MMP1MMP13MMP9
SCHEMBL6562064 0.81 ADAM17 (0.43) KEAP1NFE2L2MAPTMMP1MMP13
SCHEMBL6562044 0.81 NQO2 (0.37) F2F10PRSS1
SCHEMBL6563633 0.80 NQO2 (0.37) F2F10PRSS1
SCHEMBL6563280 0.79 NQO2 (0.35) SMN1; SMN2ALDH1A1L3MBTL1F2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140802-B1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA (DE) 2004-03-17 EP disclosed
US-6479524-B1 TO PROLONG THE THROMBIN TIME BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-11-12 US disclosed
EP-1140802-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM KG (DE) 2001-10-10 EP disclosed
WO-2000035859-A1 SUBSTITUTED ARYL AND HETEROARYL DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINES BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-06-22 WO disclosed